Narcolepsy

disease
On this page

Also known as narcolepsy with or without cataplexynarcolepsy, without cataplexyparoxysmal sleep

Summary

Narcolepsy (MONDO:0021107) is a disease with 6 GWAS associations across 4 studies and 102 clinical trials. Top therapeutic interventions include pitolisant, modafinil, and armodafinil. A subtype of sleep-wake disorder — broader associated-gene and molecular evidence is on the parent page (see Disease family below).

At a glance

  • GWAS associations: 6
  • Clinical trials: 102

Clinical features

No curated clinical features (Orphanet) for this disease.

Identifiers

Disease identifiers

FieldValue
Canonical namenarcolepsy
Mondo IDMONDO:0021107
MeSHD009290
Orphanet619284
DOIDDOID:8986
ICD-10-CMG47.41
ICD-111201727099
NCITC84489
SNOMED CT60380001
UMLSC0027404
MedGen45001
GARD0022460
Is cancer (heuristic)no

Also known as: narcolepsy with or without cataplexy · narcolepsy, without cataplexy · paroxysmal sleep

Data availability: 6 GWAS associations (4 studies).

Disease family

This is a subtype of sleep-wake disorder. Genetic, therapeutic, and trial evidence is largely curated at the broader-term level — see the parent page for the associated-gene cohort and molecular evidence.

Classification path: disease › human disease › disease by developmental or physiological process › sleep disordersleep-wake disordernarcolepsy

Related subtypes (11): bruxism, recurrent hypersomnia, sleep apnea syndrome, hypersomnia, periodic limb movement disorder, REM sleep behavior disorder, autosomal dominant cerebellar ataxia, deafness and narcolepsy, hereditary sensory neuropathy-deafness-dementia syndrome, autoimmune encephalopathy with parasomnia and obstructive sleep apnea, circadian rhythm sleep disorder, sleep disorder, initiating and maintaining sleep

Subtypes (3): narcolepsy-cataplexy syndrome, narcolepsy without cataplexy, hereditary narcolepsy

Genetics & variants

GWAS landscape

6 GWAS associations across 4 studies. Top hits map to 3 distinct genes (as reported by GWAS).

Top associations by p-value

rsIDp-valueGeneRisk alleleOdds ratio
rs92716876e-18HLA-DRB1 - HLA-DQA1A0.45
rs1852848774e-14MUC13A3.04
rs5587739557e-13DSCAMG3.4
rs1907725334e-12HSPA4 - RPL6P15A2.69
rs1483407425e-12THEMIS - PTPRKA2.86
rs5764047974e-11LPIN3G3.81

Top studies (by case count)

StudyLead authorYearCasesControlsTitle
GCST90477562Verma A20241,079449,612Diversity and scale: Genetic architecture of 2068 traits in the VA Million Veteran Program.
GCST90480022Verma A2024414121,317Diversity and scale: Genetic architecture of 2068 traits in the VA Million Veteran Program.
GCST90481880Verma A2024414121,317Diversity and scale: Genetic architecture of 2068 traits in the VA Million Veteran Program.
GCST007779Hallberg P2019414,891Pandemrix-induced narcolepsy is associated with genes related to immunity and neuronal survival.

Variant details and genetic-evidence tiers

Tier distribution (top 50 variants)

TierVariants
Tier 1: coding0
Tier 2: splice/UTR1
Tier 3: regulatory0
Tier 4: intronic/intergenic5

MAF distribution

BucketVariants
common (>=0.05)1
low_freq (0.01-0.05)0
rare (<0.01)5
unknown0

Functional consequences

ConsequenceCount
intergenic_variant4
intron_variant1
3_prime_UTR_variant1

Top variants

rsIDChrPosAllelesMAFConsequenceGenep-valueTier
rs9271687632625208A>G,T0.162intergenic_variantHLA-DRB1 - HLA-DQA16e-18Tier 4: intronic/intergenic
rs1852848773124943465A>C0.001intergenic_variantMUC134e-14Tier 4: intronic/intergenic
rs5587739552140665321G>A,C0.001intron_variantDSCAM7e-13Tier 4: intronic/intergenic
rs1907725335133143182A>G0.001intergenic_variantHSPA4 - RPL6P154e-12Tier 4: intronic/intergenic
rs1483407426127942572A>G0.001intergenic_variantTHEMIS - PTPRK5e-12Tier 4: intronic/intergenic
rs5764047972041359205G>A03_prime_UTR_variantLPIN34e-11Tier 2: splice/UTR

Genes & proteins

No associated-gene cohort resolved for this disease. Atlas builds the molecular and therapeutic sections — associated genes, protein families, druggability, pathways, interactions, and drug associations — by aggregating over a disease’s associated genes (resolved via GWAS / GenCC / ClinVar / CIViC), and none resolved here. This is expected for antibody-mediated, autoimmune, or otherwise non-gene-defined conditions; the curated evidence for this disease is its clinical features, GWAS susceptibility, and clinical trials (above).

Function

No pathway enrichment — requires an associated-gene cohort.

Therapeutics

Drugs indicated for this disease

4 approved, 2 in late-stage (phase 3) trials. Disease-direct ChEMBL indications, not inferred from the associated-gene cohort below.

DrugDevelopment status
ArmodafinilApproved (phase 4)
DextroamphetamineApproved (phase 4)
MethylphenidateApproved (phase 4)
ModafinilApproved (phase 4)
PitolisantPhase 3 (in late-stage trials)
SolriamfetolPhase 3 (in late-stage trials)

Earlier-phase candidates (phase 2, investigational — efficacy not yet established): Clarithromycin, Mazindol.

Clinical trials & evidence

Clinical trials

Clinical trials: 102.

Phase distribution (across all retrieved trials)

PhaseTrials
Not specified49
PHASE321
PHASE214
PHASE113
PHASE43
PHASE1/PHASE21
EARLY_PHASE11

Top trials by phase / activity

NCTPhaseStatusTitle
NCT04794491PHASE4COMPLETEDAn Interventional Safety Switch Study (Segue Study) of XYWAV in Narcolepsy
NCT05869773PHASE4COMPLETEDA Switch Study From High-Sodium Oxybate to Xywav to Evaluate Changes in Blood Pressure in Participants With Narcolepsy
NCT05875974PHASE4COMPLETEDA Study to Investigate the Effect of XYWAV on Sleepiness, Polysomnography, and Functional Outcomes in Participants With Idiopathic Hypersomnia or Narcolepsy
NCT07540364PHASE3NOT_YET_RECRUITINGA Phase 3 Study to Evaluate the Efficacy and Safety of Samelisant in Patients With Narcolepsy
NCT00049803PHASE3COMPLETEDSafety and Efficacy of Xyrem Oral Solution (Sodium Oxybate) Compared With Placebo in Narcoleptic Patients
NCT00066170PHASE3COMPLETEDTrial Comparing Effects of Xyrem Taken Orally and Modafinil With Placebo in Treating Daytime Sleepiness in Narcolepsy
NCT00078312PHASE3COMPLETEDArmodafinil (CEP-10953) for Treatment of Narcolepsy, Obstructive Sleep Apnea/Hypopnea Syndrome, or Chronic Shift Work Sleep Disorder
NCT00078377PHASE3COMPLETEDSafety and Efficacy Study of Armodafinil (CEP-10953) in the Treatment of Excessive Sleepiness Associated With Narcolepsy
NCT00107796PHASE3COMPLETEDStudy of PROVIGIL ® (Modafinil) Treatment in Children and Adolescents With Excessive Sleepiness Associated With Narcolepsy
NCT00107848PHASE3COMPLETEDPROVIGIL® (Modafinil) Treatment in Children and Adolescents With Excessive Sleepiness Associated With Narcolepsy or Obstructive Sleep Apnea/Hypopnea Syndrome
NCT00132873PHASE3COMPLETEDTrial of Xyrem® (Sodium Oxybate) for the Treatment of Narcolepsy
NCT00214968PHASE3COMPLETEDAssess the Safety and Effectiveness of PROVIGIL Treatment in Children and Adolescents With Excessive Sleepiness
NCT00228553PHASE3COMPLETEDExtension Study of the Safety and Efficacy of Armodafinil in the Treatment of Patients With Excessive Sleepiness
NCT00228566PHASE3COMPLETEDStudy to Assess Patient Reported Outcomes With Armodafinil Treatment for Excessive Sleepiness in Adults With Narcolepsy or Obstructive Sleep Apnea/Hypopnea Syndrome
NCT01067222PHASE3COMPLETEDEfficacy and Safety Study of BF2.649 in the Treatment of Excessive Daytime Sleepiness in Narcolepsy
NCT01067235PHASE3COMPLETEDEfficacy and Safety Study of BF2.649 and BF2.649 Add on Modafinil on Cataplexy in Patients With Narcolespy
NCT01399606PHASE3COMPLETEDLong Term Open Label Study in Narcolepsy With BF2.649 (Pitolisant)
NCT01789398PHASE3COMPLETEDPatient Narcoleptic Treated With BF2.649 (Pitolisant) in add-on to Sodium Oxybate (HARMONY IV)
NCT02348593PHASE3COMPLETEDTwelve-week Study of the Safety and Efficacy of JZP-110 in the Treatment of Excessive Sleepiness in Narcolepsy
NCT02348632PHASE3COMPLETEDA Long-Term Safety Study of JZP-110 in the Treatment of Excessive Sleepiness in Subjects With Narcolepsy or OSA
NCT02720744PHASE3COMPLETEDOnce-Nightly Sodium Oxybate for Treatment of Excessive Daytime Sleepiness and Cataplexy in Narcolepsy
NCT04451668PHASE3COMPLETEDAn Open Label Study of FT218 in Subjects With Narcolepsy
NCT05059223PHASE3COMPLETEDA Study to Assess the Efficacy and Safety of AXS-12 (Reboxetine) in Patients With Narcolepsy
NCT05113745PHASE3COMPLETEDA Study to Assess the Long-term Efficacy and Safety of AXS-12 (Reboxetine) in Subjects With Narcolepsy (ENCORE)
NCT07493265PHASE2RECRUITINGA Study to Evaluate the Efficacy and Safety of E2086 in Adults With Narcolepsy
NCT00366080PHASE2TERMINATEDEffectiveness Of The Drug GSK189254 In Treating Patients With Narcolepsy
NCT00424931PHASE2COMPLETEDA Safety and Effectiveness Study of a Single Dose of JNJ-17216498 in Patients With Narcolepsy
NCT01006122PHASE2COMPLETEDA Study Of A Novel Compound For Excessive Daytime Sleepiness Associated With Narcolepsy
NCT01146600PHASE2COMPLETEDClarithromycin for the Treatment of Hypersomnia
NCT01485770PHASE2COMPLETEDA Study of the Safety and Effectiveness of ADX-N05 in the Treatment of Excessive Daytime Sleepiness
NCT01681121PHASE2COMPLETEDA Study of the Safety and Effectiveness of ADX-N05 for Excessive Daytime Sleepiness in Subjects With Narcolepsy
NCT02806908PHASE2COMPLETEDStudy Assessing Effects of JZP-110 on Driving Performance in the Treatment of Excessive Sleepiness in Narcolepsy
NCT02821715PHASE2COMPLETEDSafety and Efficacy of THN102 on Sleepiness in Narcoleptic Patients
NCT02832336PHASE1/PHASE2COMPLETEDThe Effect of Caffeine on the Narcoleptic Patients
NCT03267303PHASE2COMPLETEDA Study to Evaluate the Safety and Efficacy of TS-091 in Patients with Narcolepsy
NCT03881852PHASE2COMPLETEDClinical Outcomes in Narcolepsy and Cataplexy: An Evaluation of Reboxetine Treatment (CONCERT)
NCT04072380PHASE2COMPLETEDA Study to Evaluate Safety, and Efficacy of SUVN-G3031 (Samelisant) in Patients With Narcolepsy With and Without Cataplexy
NCT04923594PHASE2COMPLETEDFour-week Study of the Safety and Efficacy of NLS-2 (Mazindol Extended Release) in the Treatment of Narcolepsy
NCT05055024PHASE2COMPLETEDAn Open Label Study of NLS-2 (Mazindol Extended Release) in Subjects With Narcolepsy
NCT07613710PHASE1RECRUITINGA Trial to Test the Safety and Tolerability of Lu AH69593 in Adults That Are Healthy or Have Narcolepsy

Drugs tested across these trials (top 30)

MoleculeMax phaseTrials referencing
PITOLISANT415
MODAFINIL411
ARMODAFINIL46
OXYBATE45
SOLRIAMFETOL44
CAFFEINE41
DEXTROAMPHETAMINE41
MAZINDOL41
SUVN-G303123
DANAVOREXTON21
GSK18925421
JNJ-1721649821
PF-0365474621