SCHEMBL28293058

SCHEMBL28293058

CC/C(=C\c1ccccc1)CO

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.52
KDM1A O60341 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
AKR1C3 P42330 1/20 0.42
NR1I2 O75469 1/20 0.42
LMNA P02545 1/20 0.41
RECQL P46063 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
FBP1 P09467 1/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
AKR1C1 Q04828 1/20 0.36
ESR1 P03372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28472907 1.00 TRPA1 (0.52) TRPA1KDM1AMEN1KMT2AALDH1A1
SCHEMBL59713 0.89 KDM1A (0.48) TRPA1KDM1AMEN1KMT2AALDH1A1
SCHEMBL216869 0.86 TSHR (0.43) TRPA1MEN1KMT2AALDH1A1TSHR
SCHEMBL1758410 0.81 CYP2A6 (0.38) TRPA1LMNARECQLTDP1ESR1
SCHEMBL11908074 0.81 CYP2A6 (0.38) TRPA1LMNARECQLTDP1ESR1
SCHEMBL17329401 0.81 KDM1A (0.47) TRPA1KDM1AMEN1KMT2AALDH1A1
SCHEMBL9312061 0.81 LMNA (0.47) TRPA1KDM1AMEN1KMT2AALDH1A1
SCHEMBL7304675 0.81 NR1I2 (0.44) TRPA1KDM1AMEN1KMT2AALDH1A1
SCHEMBL7304680 0.81 NR1I2 (0.44) TRPA1KDM1AMEN1KMT2AALDH1A1
SCHEMBL2244765 0.80 LMNA (0.44) TRPA1KDM1AMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109863137-B LSD1 inhibitors and medical uses thereof 星座制药公司 2022-12-16 CN disclosed
CN-109863137-A LSD1 inhibitor and its medical usage 星座制药公司 2019-06-07 CN disclosed