SCHEMBL3662631

SCHEMBL3662631

CN(CCC1CCCc2c1cnn2C)C1CCCCC1.CN(CCC1CCCc2c1cnn2C)Cc1ccccc1.Cn1ncc2c1CCCC2CCN1CCC(O)(c2ccccc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.50
TMEM97 Q5BJF2 1/20 0.40
OPRL1 P41146 2/20 0.34
DRD2 P14416 3/20 0.34
HTR1A P08908 2/20 0.34
HTR2A P28223 2/20 0.34
POLB P06746 1/20 0.33
DRD1 P21728 1/20 0.32
DRD5 P21918 1/20 0.32
HRH1 P35367 1/20 0.32
DRD3 P35462 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL956233 0.85 SIGMAR1 (0.67) SIGMAR1TMEM97OPRL1DRD2HTR1A
SCHEMBL954722 0.80 SIGMAR1 (0.58) SIGMAR1TMEM97DRD2HTR1AHTR2A
SCHEMBL5170674 0.79 SIGMAR1 (0.80) SIGMAR1TMEM97DRD2HTR1AHTR2A
Oxalic Acid SCHEMBL956463 0.78 SIGMAR1 (0.53) SIGMAR1TMEM97
SCHEMBL957063 0.76 SIGMAR1 (0.51) SIGMAR1TMEM97DRD2HTR1AHTR2A
SCHEMBL2332817 0.73 SIGMAR1 (0.57) SIGMAR1TMEM97DRD2HTR1AHTR2A
SCHEMBL956607 0.71 SIGMAR1 (0.44) SIGMAR1TMEM97POLBHRH3
Oxalic Acid SCHEMBL3567521 0.71 SIGMAR1 (0.60) SIGMAR1TMEM97OPRL1DRD2HTR1A
SCHEMBL8272461 0.71 SIGMAR1 (0.48) SIGMAR1TMEM97HTR1A
SCHEMBL958098 0.70 SIGMAR1 (0.57) SIGMAR1TMEM97HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7829559-B2 Substituted pyrazole sigma receptor antagonists LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2010-11-09 US claimed