SCHEMBL6134778

SCHEMBL6134778

CCCCCS(=O)(=O)NC(=O)c1ccc2[nH]c(C)c(Cc3ccc(COc4ccccc4)cc3Cl)c2c1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 12/20 0.41
PPARG P37231 2/20 0.41
POLB P06746 3/20 0.41
PTPN1 P18031 1/20 0.41
PTPN5 P54829 1/20 0.40
CNR1 P21554 1/20 0.39
BCL2L1 Q07817 3/20 0.38
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5882026 0.88 POLB (0.50) MCL1POLBPTPN1PTPN5MAPT
SCHEMBL6134732 0.86 MAPT (0.44) MCL1PPARGPOLBPTPN5MAPT
SCHEMBL5881755 0.86 PTPN1 (0.48) MCL1PPARGPTPN1CNR1BCL2L1
SCHEMBL5882152 0.86 MAPT (0.49) MCL1PPARGPOLBPTPN1PTPN5
SCHEMBL6321321 0.85 PPARG (0.42) MCL1PPARGPOLBPTPN1PTPN5
SCHEMBL6318663 0.85 SCN9A (0.40) MCL1PPARGPOLBPTPN1PTPN5
SCHEMBL5881578 0.85 PPARG (0.55) MCL1PPARGCNR1MAPT
SCHEMBL6328588 0.85 MCL1 (0.49) MCL1POLBPTPN5BCL2L1
SCHEMBL5881778 0.85 PPARG (0.43) MCL1PPARGPTPN1PTPN5CNR1
SCHEMBL5881774 0.85 PPARG (0.43) MCL1PPARGPTPN1PTPN5CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050171185-A1 Indole derivatives FUJISAWA PHARMACEUTICAL CO., LTD., A JAPANESE CORPORATION 2005-08-04 US claimed
EP-1070705-A1 INDOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-01-24 EP claimed
WO-2005082414-A2 CONCOMITANT DRUGS OF A SULFONAMIDE AND ANOTHER THERAPEUTIC AGENT ASTELLAS PHARMA INC. (JP) 2005-09-09 WO disclosed
US-20050197376-A1 Concomitant drugs FUJISAWA PHARMACEUTICAL CO. LTD. (JP) 2005-09-08 US disclosed
US-20050171185-A1 Indole derivatives FUJISAWA PHARMACEUTICAL CO., LTD., A JAPANESE CORPORATION 2005-08-04 US disclosed
EP-1070705-A1 INDOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-01-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050171185-A1 Indole derivatives PDE5A, IGFBP5, HTR5A MCL1 3761/4885PPARG 2279/4885POLB 3673/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.