SCHEMBL7461997

SCHEMBL7461997

COc1c(N2CC[C@H](CNC3CC3)C2)c(F)c(N)c2c(=O)c(OC(=O)O)cn([C@@H]3C[C@@H]3F)c12

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.40
CYP3A4 P08684 1/20 0.38
TOP1 P11387 9/20 0.36
GSK3B P49841 4/20 0.34
CACNA1F O60840 1/20 0.33
POLB P06746 1/20 0.33
MAPK1 P28482 1/20 0.33
CACNA1D Q01668 1/20 0.33
CACNA1S Q13698 1/20 0.33
CACNA1C Q13936 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7462916 0.91 KCNH2 (0.34) KCNH2CYP3A4TOP1CACNA1FPOLB
SCHEMBL7463545 0.90 KCNH2 (0.48) KCNH2CYP3A4TOP1GSK3BCACNA1F
SCHEMBL7468912 0.90 KCNH2 (0.48) KCNH2CYP3A4TOP1GSK3BCACNA1F
SCHEMBL15062970 0.89 CYP3A4 (0.35) KCNH2CYP3A4TOP1GSK3BCACNA1F
SCHEMBL15063054 0.82 KCNH2 (0.42) KCNH2GSK3BCACNA1FPOLBMAPK1
SCHEMBL15063038 0.80 CACNA1F (0.36) KCNH2CYP3A4GSK3BCACNA1FPOLB
SCHEMBL7467420 0.79 KCNH2 (0.46) KCNH2CYP3A4GSK3BCACNA1FPOLB
Hydrochloric Acid SCHEMBL7468673 0.79 KCNH2 (0.45) KCNH2CYP3A4GSK3BCACNA1FPOLB
SCHEMBL7461815 0.79 KCNH2 (0.43) KCNH2CYP3A4TOP1POLB
SCHEMBL500422 0.78 KCNH2 (0.46) KCNH2CYP3A4GSK3BCACNA1FPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900793-B1 CYCLOALKYLAMINOMETHYLPYRROLIDINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2002-07-24 EP claimed