SCHEMBL7679588

SCHEMBL7679588

O=COc1c(OCC2CO2)ccc2occc12

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
GLA P06280 1/20 0.38
HTR2C P28335 15/20 0.37
HTR2A P28223 12/20 0.37
HTR2B P41595 11/20 0.37
TDP1 Q9NUW8 1/20 0.35
TP53 P04637 1/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HIF1A Q16665 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
PKM P14618 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6195483 0.84 ALDH1A1 (0.40) ALDH1A1GLAHTR2CHTR2AHTR2B
SCHEMBL23552017 0.79 TDP1 (0.36) ALDH1A1GLAHTR2CHTR2AHTR2B
SCHEMBL6975228 0.75 ALDH1A1 (0.41) ALDH1A1GLAHTR2ATDP1TP53
SCHEMBL6975232 0.75 ALDH1A1 (0.41) ALDH1A1GLAHTR2ATDP1TP53
SCHEMBL6309690 0.74 ALDH1A1 (0.53) ALDH1A1GLAHTR2CHTR2AHTR2B
SCHEMBL6309685 0.74 ALDH1A1 (0.53) ALDH1A1GLAHTR2CHTR2AHTR2B
SCHEMBL7966131 0.74 ALDH1A1 (0.53) ALDH1A1GLAHTR2CHTR2AHTR2B
SCHEMBL6985499 0.72 ALDH1A1 (0.48) ALDH1A1GLATDP1TP53CYP3A4
SCHEMBL6985498 0.72 ALDH1A1 (0.48) ALDH1A1GLATDP1TP53CYP3A4
SCHEMBL6978043 0.72 ALDH1A1 (0.48) ALDH1A1GLATDP1TP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6353002-B2 DIOXINOINDOLE AND THIENOBENZODIOXIN COMPOUNDS WHICH ARE HT3 RECEPTOR ANTAGONISTS AND ARE USED TO TREAT CENTRAL NERVOUS SYSTEM DISORDERS KNOLL AKTIENGESELLSCHAFT (DE) 2002-03-05 US disclosed
US-20010008903-A1 Therapeutic agents BIRCH ALAN MARTIN (GB) 2001-07-19 US disclosed
US-6201004-B1 CENTRAL NERVOUS SYSTEM, PSYCHOLOGICAL, EATING, CARDIOVASCULAR, BRAIN, AND GASTROINTESTINAL DISORDERS KNOLL AKTIENGESELLSCHAFT (DE) 2001-03-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010008903-A1 Therapeutic agents GPR119, SNCA, HTR2B ALDH1A1 3243/4885GLA 601/4885HTR2C 7/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.