SCHEMBL8534985

SCHEMBL8534985

Cc1c(-c2ccc(Cc3ccc(OC(F)(F)F)cc3)cc2)n(O)c2cc(Cl)ccc2c1=O

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 2/20 0.40
CYP3A4 P08684 1/20 0.40
PTGDR2 Q9Y5Y4 2/20 0.39
ESR1 P03372 3/20 0.38
DHODH Q02127 1/20 0.37
MAPK9 P45984 1/20 0.37
TRPC5 Q9UL62 1/20 0.36
SERPINE1 P05121 2/20 0.36
OPRK1 P41145 1/20 0.36
GRM2 Q14416 1/20 0.36
PPARG P37231 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
PTGES O14684 1/20 0.35
DDR1 Q08345 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8535025 0.85 ESR1 (0.39) ESR1SERPINE1GRM2PPARG
SCHEMBL8535303 0.76 MAT2A (0.55) CYP3A4PTGDR2
SCHEMBL8534631 0.76 PPARG (0.40) SERPINE1PPARG
SCHEMBL29240187 0.74 ALDH1A1 (0.51) MAPK8CYP3A4MAPK9PPARG
SCHEMBL30866017 0.71 ESR1 (0.43) MAPK8ESR1MAPK9
SCHEMBL29240230 0.71 ESR1 (0.44) ESR1PPARGTRPV1
SCHEMBL29240188 0.71 ESR1 (0.43) MAPK8ESR1MAPK9
SCHEMBL30866019 0.71 ESR1 (0.44) ESR1PPARGTRPV1
SCHEMBL8532926 0.70 MAT2A (0.51) CYP3A4
SCHEMBL8514142 0.69 ALOX5 (0.48) OPRK1PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO claimed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed