SCHEMBL8555310

SCHEMBL8555310

NCC(=O)c1csc2cccnc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 6/20 0.44
LIMK1 P53667 1/20 0.41
PARP1 P09874 1/20 0.38
IRAK1 P51617 3/20 0.38
SYK P43405 2/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 4/20 0.35
HSD17B10 Q99714 1/20 0.35
ALOX15 P16050 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NAPRT Q6XQN6 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30844941 0.82 PARP1 (0.53) IRAK4LIMK1PARP1IRAK1KDM4E
SCHEMBL19555042 0.82 PARP1 (0.53) IRAK4LIMK1PARP1IRAK1KDM4E
Hydrochloric Acid SCHEMBL30845090 0.81 PARP1 (0.51) IRAK4LIMK1PARP1IRAK1KDM4E
SCHEMBL29560247 0.80 KDM4E (0.48) IRAK4LIMK1IRAK1KDM4EALDH1A1
SCHEMBL7114666 0.80 KDM4E (0.48) IRAK4LIMK1IRAK1KDM4EALDH1A1
SCHEMBL17023631 0.79 IRAK4 (0.49) IRAK4LIMK1PARP1IRAK1SYK
SCHEMBL30845404 0.75 IRAK4 (0.55) IRAK4LIMK1IRAK1SYKKDM4E
SCHEMBL8597003 0.75 IKBKB (0.41) LIMK1KDM4EALDH1A1HSD17B10NAPRT
SCHEMBL8440763 0.75 TDP1 (0.43) IRAK4LIMK1ALDH1A1HDAC3HDAC4
Trifluoroacetic Acid SCHEMBL30844916 0.74 L3MBTL1 (0.50) IRAK4LIMK1PARP1IRAK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0581106-B1 Substituted aminothienopyridines, a process for their preparation and their use as medicaments HOECHST MARION ROUSSEL INC (US) 1998-05-20 EP disclosed