SCHEMBL8998932

SCHEMBL8998932

CC(C#N)(SSC(C)(C#N)c1c[nH]c2ccccc12)c1c[nH]c2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 2/20 0.46
IMPDH1 P20839 1/20 0.46
APP P05067 1/20 0.43
ATM Q13315 1/20 0.42
CYP2A6 P11509 1/20 0.39
POLB P06746 1/20 0.38
GPR84 Q9NQS5 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
MAPT P10636 2/20 0.37
CYP3A4 P08684 1/20 0.37
AHR P35869 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
FFAR1 O14842 1/20 0.37
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
TUBA1B P68363 1/20 0.37
TUBA4A P68366 1/20 0.37
TUBB4B P68371 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8999076 0.90 IMPDH2 (0.46) IMPDH2IMPDH1APPATMCYP2A6
SCHEMBL997167 0.83 IMPDH2 (0.52) IMPDH2IMPDH1APPATMCYP2A6
SCHEMBL9593180 0.81 IMPDH2 (0.50) IMPDH2IMPDH1APPATMCYP2A6
SCHEMBL11797189 0.75 ATM (0.50) IMPDH2IMPDH1ATMCYP2A6GPR84
SCHEMBL799601 0.75 ATM (0.54) IMPDH2IMPDH1ATMCYP2A6GPR84
SCHEMBL29885789 0.75 ATM (0.54) IMPDH2IMPDH1ATMCYP2A6GPR84
SCHEMBL13335152 0.75 ATM (0.54) IMPDH2IMPDH1ATMCYP2A6GPR84
SCHEMBL30437029 0.75 ATM (0.54) IMPDH2IMPDH1ATMCYP2A6GPR84
SCHEMBL1685393 0.75 ATM (0.54) IMPDH2IMPDH1ATMCYP2A6GPR84
SCHEMBL23478771 0.73 ATM (0.47) IMPDH2IMPDH1ATMCYP2A6GPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5556874-A ENZYME INHIBITORS AS ANTICARCINOGENIC AGENTS WARNER LAMBERT COMPANY (US) 1996-09-17 US disclosed
US-5464861-A Anticarcinogenic agents WARNER-LAMBERT (US) 1995-11-07 US disclosed
EP-0654024-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1995-05-24 EP disclosed
WO-1994003427-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1994-02-17 WO disclosed