SCHEMBL10053271

SCHEMBL10053271

CCN(C)Cc1cccc(B2OCc3cc(F)ccc32)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
PDE3A Q14432 1/20 0.41
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
MEN1 O00255 5/20 0.33
KMT2A Q03164 5/20 0.33
NPC1 O15118 1/20 0.33
RIPK1 Q13546 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRL1 P41146 1/20 0.32
ACHE P22303 2/20 0.31
SLC6A3 Q01959 1/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
TSPO P30536 1/20 0.31
PYCR1 P32322 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10053174 0.91 CA1 (0.41) CA1CA2PDE3AACHEPDE4A
SCHEMBL10053172 0.91 CA1 (0.43) CA1CA2PDE3AMEN1KMT2A
SCHEMBL10053144 0.87 CA1 (0.46) CA1CA2PDE3APDE4APDE4B
SCHEMBL10053152 0.86 MEN1 (0.41) CA1CA2PDE3AMEN1KMT2A
SCHEMBL10053184 0.84 CA1 (0.36) CA1CA2PDE3AMEN1KMT2A
SCHEMBL597009 0.82 CA1 (0.49) CA1CA2PDE3APDE4APDE4B
SCHEMBL12589683 0.82 CA1 (0.46) CA1CA2PDE3APDE4APDE4B
SCHEMBL10077708 0.81 CA1 (0.43) CA1CA2PDE3ACHRNB2CHRNA4
SCHEMBL10077714 0.81 CA1 (0.40) CA1CA2PDE3APDE4APDE4B
SCHEMBL10053160 0.80 CA1 (0.47) CA1CA2PDE3ASLC6A3PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106031-B2 Hydrolytically-resistant boron-containing therapeutics and methods of use ANACOR PHARMACEUTICALS, INC. (US) 2012-01-31 US disclosed