SCHEMBL10053274

SCHEMBL10053274

CCc1cc(B2OCc3cc(F)ccc32)ccc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
PDE3A Q14432 1/20 0.43
HTR2A P28223 1/20 0.36
SLC6A4 P31645 1/20 0.36
KCNH2 Q12809 1/20 0.36
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
P2RX7 Q99572 1/20 0.32
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
MAPT P10636 1/20 0.30
CYP2C9 P11712 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10053162 0.88 CA1 (0.47) CA1CA2PDE3APDE4APDE4B
SCHEMBL10053178 0.81 CA1 (0.47) CA1CA2PDE3APDE4APDE4B
SCHEMBL10053161 0.80 CA1 (0.49) CA1CA2PDE3AKCNH2PDE4A
SCHEMBL10053151 0.80 CA1 (0.47) CA1CA2PDE3APDE4APDE4B
SCHEMBL10053170 0.80 CA1 (0.41) CA1CA2PDE3AHTR2ASLC6A4
SCHEMBL10053182 0.79 CA1 (0.61) CA1CA2PDE3APDE4APDE4B
SCHEMBL10053279 0.79 CA1 (0.50) CA1CA2PDE3APDE4APDE4B
SCHEMBL500198 0.78 CA1 (0.59) CA1CA2PDE3APDE4APDE4B
SCHEMBL10053272 0.78 CA1 (0.47) CA1CA2PDE3APDE4APDE4B
SCHEMBL10053144 0.77 CA1 (0.46) CA1CA2PDE3APDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106031-B2 Hydrolytically-resistant boron-containing therapeutics and methods of use ANACOR PHARMACEUTICALS, INC. (US) 2012-01-31 US disclosed