SCHEMBL10053285

SCHEMBL10053285

Cc1cncc(B2OCc3cc(F)ccc32)c1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
PDE3A Q14432 1/20 0.48
PDE4A P27815 2/20 0.35
PDE4B Q07343 2/20 0.35
PDE4C Q08493 2/20 0.35
PDE4D Q08499 2/20 0.35
TDO2 P48775 1/20 0.34
CYP11B1 P15538 4/20 0.32
CYP11B2 P19099 4/20 0.32
GPR55 Q9Y2T6 1/20 0.31
ADRA2A P08913 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30
ADRA1B P35368 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10053169 0.85 CA1 (0.53) CA1CA2PDE3APDE4APDE4B
SCHEMBL500011 0.84 CA1 (0.49) CA1CA2PDE3APDE4APDE4B
SCHEMBL10053194 0.83 CA1 (0.48) CA1CA2PDE3APDE4APDE4B
SCHEMBL500871 0.82 CA1 (0.53) CA1CA2PDE3APDE4APDE4B
SCHEMBL500067 0.82 CA1 (0.49) CA1CA2PDE3APDE4APDE4B
SCHEMBL10053182 0.80 CA1 (0.61) CA1CA2PDE3APDE4APDE4B
SCHEMBL10053279 0.80 CA1 (0.50) CA1CA2PDE3APDE4APDE4B
SCHEMBL500198 0.79 CA1 (0.59) CA1CA2PDE3APDE4APDE4B
SCHEMBL500789 0.78 CA1 (0.54) CA1CA2PDE3APDE4APDE4B
SCHEMBL10053178 0.77 CA1 (0.47) CA1CA2PDE3APDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106031-B2 Hydrolytically-resistant boron-containing therapeutics and methods of use ANACOR PHARMACEUTICALS, INC. (US) 2012-01-31 US disclosed