SCHEMBL10054022

SCHEMBL10054022

Bc1ccc(/C=C/c2ccc(N(c3ccc(C)cc3)c3ccc(C(C)(C)C)cc3)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
PTGS1 P23219 2/20 0.41
PTGS2 P35354 2/20 0.41
CYP1A2 P05177 2/20 0.40
NFE2L2 Q16236 4/20 0.38
HCRTR2 O43614 1/20 0.38
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
RELA Q04206 1/20 0.36
RAB9A P51151 4/20 0.35
NPC1 O15118 3/20 0.35
MAPT P10636 3/20 0.35
ALOX5 P09917 1/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
APOBEC3A P31941 2/20 0.34
APOBEC3G Q9HC16 2/20 0.34
CYP1A1 P04798 1/20 0.33
CYP1B1 Q16678 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13045361 1.00 TSHR (0.47) TSHRPTGS1PTGS2CYP1A2NFE2L2
SCHEMBL13892093 0.94 CYP1A2 (0.44) TSHRCYP1A2NR1H2NR1H3RELA
SCHEMBL14424330 0.92 TSHR (0.56) TSHRPTGS1PTGS2CYP1A2NFE2L2
SCHEMBL13636796 0.92 TSHR (0.56) TSHRPTGS1PTGS2CYP1A2NFE2L2
SCHEMBL13636804 0.92 TSHR (0.56) TSHRPTGS1PTGS2CYP1A2NFE2L2
SCHEMBL9604060 0.92 TSHR (0.56) TSHRPTGS1PTGS2CYP1A2NFE2L2
SCHEMBL13358630 0.87 TSHR (0.50) TSHRPTGS1PTGS2CYP1A2NFE2L2
SCHEMBL13358765 0.87 TSHR (0.50) TSHRPTGS1PTGS2CYP1A2NFE2L2
SCHEMBL10054025 0.86 CYP1A2 (0.39) CYP1A2NR1H2NR1H3RELARAB9A
SCHEMBL14508552 0.86 CYP1A2 (0.39) CYP1A2NR1H2NR1H3RELARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012013310-A1 POLYMERS CONTAINING SUBSTITUTED BENZODITHIOPHENE UNITS, BLENDS CONTAINING SAID POLYMERS, AND DEVICES CONTAINING SAID POLYMERS OR BLENDS MERCK PATENT GMBH (DE) 2012-02-02 WO disclosed