SCHEMBL10069049

SCHEMBL10069049

COCCOc1cc(C(=O)OC)cc(C(OC(=N)C(Cl)(Cl)Cl)c2cccc(F)c2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.40
AURKA O14965 1/20 0.38
RPS6KB1 P23443 1/20 0.38
LMNA P02545 3/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
MAPT P10636 3/20 0.34
RAB9A P51151 3/20 0.34
NPC1 O15118 2/20 0.34
REN P00797 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
PLA2G4A P47712 1/20 0.34
GCK P35557 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
SLC6A9 P48067 1/20 0.33
SLC6A5 Q9Y345 1/20 0.33
CNR2 P34972 1/20 0.33
ROCK2 O75116 1/20 0.33
HTR1A P08908 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10069048 0.81 MRGPRX4 (0.44) MRGPRX4AURKARPS6KB1LMNAMEN1
SCHEMBL10069050 0.80 AURKA (0.40) MRGPRX4AURKARPS6KB1LMNAMEN1
SCHEMBL10069061 0.72 KMT2A (0.56) MRGPRX4LMNAMEN1KMT2AMAPT
SCHEMBL10068778 0.71 HPGD (0.43) MEN1KMT2AMAPTRAB9AALDH1A1
SCHEMBL10068802 0.70 KLKB1 (0.41) LMNAMEN1KMT2AMAPTRAB9A
SCHEMBL10069568 0.69 MEN1 (0.48) MEN1KMT2AMAPTNPC1ALDH1A1
SCHEMBL38987 0.68 MAPT (0.59) LMNAMAPTRAB9AALDH1A1GAA
SCHEMBL2809253 0.68 MAPT (0.59) LMNAMAPTRAB9ANPC1ALDH1A1
SCHEMBL10068957 0.66 HPGD (0.42) MAPTALDH1A1GAAPLA2G4A
SCHEMBL10068953 0.66 KLKB1 (0.40) LMNAMEN1KMT2AMAPTREN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012019428-A1 BENZOHYDROL DERIVATIVES, A PREPARATION PROCESS AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-02-16 WO disclosed