SCHEMBL10072096

SCHEMBL10072096

CC(C)COC(C)ONC(=O)/C=C/c1ccc(CNC2(C(=O)OC3CCCC3)CC2)nc1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAP3K7 O43318 2/20 0.34
TAB1 Q15750 2/20 0.34
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC4 P56524 1/20 0.30
MEF2D Q14814 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10072275 0.98 MAP3K7 (0.33) MAP3K7TAB1NPC1RAB9ASMN1; SMN2
SCHEMBL10072098 0.95 MAP3K7 (0.32) MAP3K7TAB1NPC1RAB9ASMN1; SMN2
SCHEMBL7897506 0.88 SMN1; SMN2 (0.38) NPC1RAB9ASMN1; SMN2HDAC1HDAC4
SCHEMBL9895879 0.88 SMN1; SMN2 (0.38) NPC1RAB9ASMN1; SMN2HDAC1HDAC4
SCHEMBL9895162 0.85 HDAC3 (0.39) NPC1RAB9ASMN1; SMN2HDAC1HDAC4
SCHEMBL7896386 0.85 HDAC3 (0.39) NPC1RAB9ASMN1; SMN2HDAC1HDAC4
SCHEMBL9895415 0.83 MAP3K7 (0.30) MAP3K7TAB1
SCHEMBL10072240 0.83 SMN1; SMN2 (0.36) NPC1RAB9ASMN1; SMN2HDAC1HDAC4
SCHEMBL7899126 0.83 MAP3K7 (0.30) MAP3K7TAB1
SCHEMBL2731939 0.83 HDAC4 (0.43) HDAC1HDAC4MEF2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012025701-A1 ALPHA, ALPHA - DI SUBSTITUTED GLYCINE ESTER DERIVATIVES AND THEIR USE AS HDAC INHIBITORS CHROMA THERAPEUTICS LTD. (GB) 2012-03-01 WO disclosed