SCHEMBL10087503

SCHEMBL10087503

CCc1ccc(O)cc1I

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYR P14679 5/20 0.45
HSD17B3 P37058 1/20 0.43
MEN1 O00255 1/20 0.42
TP53 P04637 1/20 0.42
CYP3A4 P08684 1/20 0.42
ALOX5 P09917 1/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
GABRA1 P14867 1/20 0.41
GABRB2 P47870 1/20 0.41
HSP90AB1 P08238 1/20 0.41
TTR P02766 1/20 0.41
HSD17B1 P14061 1/20 0.40
ESRRB O95718 1/20 0.40
ESR1 P03372 1/20 0.40
ESRRA P11474 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4652298 0.84 HSD17B3 (0.42) TYRHSD17B3MEN1TP53CYP3A4
SCHEMBL30979257 0.80 TYR (0.48) TYRHSD17B3MEN1TP53CYP3A4
SCHEMBL1724358 0.80 TYR (0.48) TYRHSD17B3MEN1TP53CYP3A4
SCHEMBL16528479 0.78 ANPEP (0.49) TYRHSD17B3MEN1TP53CYP3A4
SCHEMBL29492456 0.78 TYR (0.65) TYRMEN1TP53CYP3A4ALOX5
SCHEMBL40375 0.78 TYR (0.65) TYRMEN1TP53CYP3A4ALOX5
SCHEMBL13019662 0.78 TTR (0.36) GABRA1GABRB2TTRTNIK
SCHEMBL9579057 0.76 TYR (0.56) TYRHSD17B3MEN1TP53CYP3A4
SCHEMBL2571546 0.76 TYR (0.45) TYRHSD17B3MEN1TP53CYP3A4
SCHEMBL16526930 0.76 MAPT (0.39) MAPTTSHRHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937666-B1 SUBSTITUTED HETEROCYCLIC COMPOUNDS WITH CXCR3 ANTAGONIST ACTIVITY SCHERING CORP (US) 2012-02-22 EP disclosed