SCHEMBL10122759

SCHEMBL10122759

CC(C)(N)CC(C(N)=O)c1ccc(Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.42
HTR2A P28223 1/20 0.42
SLC6A4 P31645 1/20 0.42
HRH1 P35367 1/20 0.42
HTR2B P41595 1/20 0.42
CHRNA4 P43681 1/20 0.42
SLC6A3 Q01959 1/20 0.42
POLB P06746 2/20 0.41
CYP2C9 P11712 4/20 0.41
CYP2C19 P33261 3/20 0.41
MEN1 O00255 2/20 0.41
CYP2D6 P10635 2/20 0.41
KMT2A Q03164 2/20 0.41
AOC3 Q16853 1/20 0.40
BRD4 O60885 1/20 0.40
GABBR2 O75899 3/20 0.39
GABBR1 Q9UBS5 3/20 0.39
LMNA P02545 2/20 0.39
CYP3A4 P08684 1/20 0.39
ADORA3 P0DMS8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12167835 1.00 SLC6A2 (0.42) SLC6A2HTR2ASLC6A4HRH1HTR2B
SCHEMBL685065 0.87 BRD4 (0.47) SLC6A2HTR2ASLC6A4HRH1HTR2B
SCHEMBL684422 0.87 BRD4 (0.47) SLC6A2HTR2ASLC6A4HRH1HTR2B
SCHEMBL684738 0.87 BRD4 (0.47) SLC6A2HTR2ASLC6A4HRH1HTR2B
SCHEMBL8919457 0.84 CYP2C9 (0.44) POLBCYP2C9CYP2C19MEN1CYP2D6
SCHEMBL680865 0.84 POLB (0.42) SLC6A2HTR2ASLC6A4HRH1HTR2B
SCHEMBL679766 0.84 POLB (0.42) SLC6A2HTR2ASLC6A4HRH1HTR2B
SCHEMBL680823 0.84 POLB (0.42) SLC6A2HTR2ASLC6A4HRH1HTR2B
SCHEMBL12167826 0.83 AOC3 (0.40) AOC3
SCHEMBL22758202 0.81 CYP2C9 (0.41) POLBCYP2C9CYP2C19MEN1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087336-A1 AUTOPHAGY INDUCER AND INHIBITOR COMBINATION THERAPY FOR THE TREATMENT OF NEOPLASMS GENENTECH, INC. (US) 2012-06-28 WO disclosed
WO-2011130654-A1 FOX03A AS PREDICTIVE BIOMARKER FOR PI3K/AKT KINASE PATHWAY INHIBITOR EFFICACY GENENTECH, INC. (US) 2011-10-20 WO disclosed