SCHEMBL10127971

SCHEMBL10127971

CCc1cc(C)cc(CC)c1C1C(=O)C2CC(CC/C(C)=N/OC)CC2C1=O

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2731711 1.00 CYP3A4 (0.34) CYP3A4CYP2D6MAPT
SCHEMBL2730222 0.83
SCHEMBL4766218 0.80 BRD4 (0.31)
SCHEMBL15641213 0.78
SCHEMBL2731712 0.77 CYP3A4 (0.33) CYP3A4CYP2D6MAPT
SCHEMBL16994571 0.73
SCHEMBL10127398 0.72
SCHEMBL16994203 0.72
SCHEMBL12885590 0.70
SCHEMBL4774264 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2635550-B1 PHENYL-SUBSTITUTED BICYCLOOCTANE-1,3-DIONE-DERIVATIVES BAYER IP GMBH (DE) 2016-01-27 EP disclosed
US-9101133-B2 Phenyl-substituted bicyclooctane-1,3-dione-derivatives BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-08-11 US disclosed
US-9101133-B2 Phenyl-substituted bicyclooctane-1,3-dione-derivatives BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-08-11 US disclosed
WO-2012059436-A2 PHENYL-SUBSTITUTED BICYCLOOCTANE-1,3-DIONE-DERIVATIVES BAYER CROPSCIENCE AG (DE) 2012-05-10 WO disclosed