SCHEMBL10129685

SCHEMBL10129685

CC(F)(F)/C=C/n1c(-c2ccc(Cl)cc2)nn(CC(=O)O)c1=O

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 10/20 0.41
AVPR1A P37288 10/20 0.41
AKR1B1 P15121 1/20 0.37
TSHR P16473 1/20 0.36
PTGDR2 Q9Y5Y4 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
MAPT P10636 1/20 0.35
CNR1 P21554 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL719971 0.91 AVPR2 (0.42) AVPR2AVPR1AAKR1B1TSHRALDH1A1
SCHEMBL256747 0.91 AVPR2 (0.42) AVPR2AVPR1AAKR1B1TSHRALDH1A1
SCHEMBL6914750 0.89 AVPR2 (0.44) AVPR2AVPR1ATSHRALDH1A1MAPT
SCHEMBL255993 0.81 AVPR2 (0.45) AVPR2AVPR1ATSHRALDH1A1MAPT
SCHEMBL21004008 0.75 AVPR2 (0.45) AVPR2AVPR1AAKR1B1TSHRALDH1A1
SCHEMBL8235255 0.75 TSHR (0.43) AVPR2AVPR1AAKR1B1TSHRALDH1A1
SCHEMBL8227129 0.75 AVPR2 (0.46) AVPR2AVPR1ATSHRPTGDR2CNR1
SCHEMBL8227138 0.75 AVPR2 (0.51) AVPR2AVPR1APTGDR2
SCHEMBL413351 0.73 AVPR2 (0.57) AVPR2AVPR1A
SCHEMBL8235257 0.73 AVPR2 (0.46) AVPR2AVPR1ATSHRPTGDR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035075-A1 SUBSTITUTED PHENYLACETATE AND PHENYLPROPANE AMIDES AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-03-22 WO disclosed