SCHEMBL1013708

SCHEMBL1013708

[CH]NC=C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17599028 0.59
SCHEMBL11129667 0.59
SCHEMBL576753 0.59
SCHEMBL10896080 0.56
SCHEMBL14398772 0.56
SCHEMBL13894520 0.56
SCHEMBL216324 0.56
SCHEMBL1330937 0.56
SCHEMBL139417 0.56
SCHEMBL3775503 0.56

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063592-B1 DIRECT PHOTOPATTERNING OF ROBUST AND DIVERSE MATERIALS CALIFORNIA INST OF TECHN (US) 2021-04-07 EP disclosed
US-10799613-B2 Direct photopatterning of robust and diverse materials CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2020-10-13 US disclosed
US-10092537-B2 Use for PAI-1 inhibitor RENASCIENCE CO., LTD. (JP) 2018-10-09 US disclosed
EP-2903996-B1 PHOTOINITIATED OLEFIN METATHESIS POLYMERIZATION CALIFORNIA INST OF TECHN (US) 2018-08-01 EP disclosed
EP-3063592-A1 DIRECT PHOTOPATTERNING OF ROBUST AND DIVERSE MATERIALS California Institute of Technology (US) 2016-09-07 EP disclosed
US-20160158188-A1 NOVEL USE FOR PAI-1 INHIBITOR RENASCIENCE CO., LTD. (JP) 2016-06-09 US disclosed
EP-2990057-A1 NOVEL USE FOR PAI-1 INHIBITOR Renascience Co., Ltd. (JP) 2016-03-02 EP disclosed
US-9207532-B2 Photoinitiated olefin methathesis polymerization CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2015-12-08 US disclosed
EP-2903996-A1 PHOTOINITIATED OLEFIN METATHESIS POLYMERIZATION California Institute of Technology (US) 2015-08-12 EP disclosed
WO-2015065649-A1 DIRECT PHOTOPATTERNING OF ROBUST AND DIVERSE MATERIALS CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2015-05-07 WO disclosed
US-20150118188-A1 DIRECT PHOTOPATTERNING OF ROBUST AND DIVERSE MATERIALS CALIFORNIA INSTITUTE OF TECHNOLOGY 2015-04-30 US disclosed
US-20140099573-A1 PHOTOINITIATED OLEFIN METHATHESIS POLYMERIZATION CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2014-04-10 US disclosed
WO-2014055720-A1 PHOTOINITIATED OLEFIN METATHESIS POLYMERIZATION CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2014-04-10 WO disclosed
US-8415479-B2 Inhibitor of plasminogen activator inhibitor-1 RENASCIENCE CO., LTD. (JP) 2013-04-09 US disclosed
US-7951806-B2 Plasminogen activator inhibitor-1 inhibitor RENASCIENCE CO., LTD. (JP) 2011-05-31 US disclosed
US-20110112140-A1 INHIBITOR OF PLASMINOGEN ACTIVATOR INHIBITOR-1 RENASCIENCE CO., LTD. (JP) 2011-05-12 US disclosed
EP-2272822-A1 INHIBITOR OF PLASMINOGEN ACTIVATOR INHIBITOR-1 Renascience CO., LTD. (JP) 2011-01-12 EP disclosed
US-20090124620-A1 PLASMINOGEN ACTIVATOR INHIBITOR-1 INHIBITOR RENASCIENCE CO., LTD. (JP) 2009-05-14 US disclosed