SCHEMBL10140906

SCHEMBL10140906

CCn1cc(C2(c3ccnc(-c4cncc(C)c4)c3)N=C(N)c3c(F)cccc32)cc(C)c1=O

nearest known ligand 0.70

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.70
KCNH2 Q12809 14/20 0.70
BACE2 Q9Y5Z0 3/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10140983 0.93 BACE1 (0.61) BACE1KCNH2BACE2
SCHEMBL9949318 0.91 BACE1 (0.81) BACE1KCNH2BACE2
SCHEMBL9949195 0.91 BACE1 (0.81) BACE1KCNH2BACE2
SCHEMBL10140391 0.89 BACE1 (0.88) BACE1KCNH2BACE2
SCHEMBL10140995 0.87 BACE1 (0.81) BACE1KCNH2BACE2
SCHEMBL9950403 0.84 BACE1 (0.67) BACE1KCNH2BACE2
SCHEMBL9948707 0.84 BACE1 (0.70) BACE1KCNH2BACE2
SCHEMBL9948853 0.83 BACE1 (0.68) BACE1KCNH2BACE2
SCHEMBL9948822 0.82 BACE1 (1.00) BACE1KCNH2BACE2
SCHEMBL9949326 0.82 BACE1 (1.00) BACE1KCNH2BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087236-A1 COMPOUNDS AND THEIR USE AS BACE INHIBITORS ASTRAZENECA AB (SE) 2012-06-28 WO disclosed