SCHEMBL10142272

SCHEMBL10142272

Cc1c(CCCC(=O)O)c2c(F)ccc(-c3ccc(OCCCCc4c(F)c(F)c(F)c(F)c4F)cc3)c2n1CCC(=O)O

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYSLTR2 Q9NS75 16/20 0.62
CYSLTR1 Q9Y271 16/20 0.62
FFAR4 Q5NUL3 4/20 0.45
FFAR1 O14842 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10142576 0.90 CYSLTR2 (0.77) CYSLTR2CYSLTR1FFAR4FFAR1
SCHEMBL10141541 0.87 CYSLTR2 (0.54) CYSLTR2CYSLTR1FFAR4FFAR1
SCHEMBL12074001 0.86 CYSLTR2 (0.68) CYSLTR2CYSLTR1FFAR4FFAR1
SCHEMBL10120784 0.85 CYSLTR2 (0.82) CYSLTR2CYSLTR1
SCHEMBL10143243 0.85 CYSLTR2 (0.76) CYSLTR2CYSLTR1
SCHEMBL597067 0.81 CYSLTR2 (0.88) CYSLTR2CYSLTR1
SCHEMBL598421 0.78 CYSLTR2 (0.77) CYSLTR2CYSLTR1
SCHEMBL12073949 0.78 CYSLTR2 (0.57) CYSLTR2CYSLTR1
SCHEMBL598114 0.77 CYSLTR2 (0.72) CYSLTR2CYSLTR1
SCHEMBL598115 0.77 CYSLTR2 (0.72) CYSLTR2CYSLTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8115014-B2 Ethynylindole compounds ONO Pharmaceuticals, Co., Ltd. (JP) 2012-02-14 US disclosed
US-20100160647-A1 ETHYNYLINDOLE COMPOUNDS ONO PHARMACEUTICAL CO., LTD. (JP) 2010-06-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100160647-A1 ETHYNYLINDOLE COMPOUNDS CYSLTR2, CYSLTR1, LTB4R2 CYSLTR2 1/4885CYSLTR1 2/4885FFAR4 246/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.