SCHEMBL10144590

SCHEMBL10144590

CNCCCn1ncc2cc(-n3ccc(-c4ccc(C(F)(F)F)cc4)cc3=O)ccc21

nearest known ligand 0.70

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 20/20 0.70
CYP3A4 P08684 2/20 0.70
CYP2C19 P33261 2/20 0.70
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10145239 0.94 MCHR1 (0.72) MCHR1CYP3A4CYP2C19
SCHEMBL538941 0.89 MCHR1 (0.75) MCHR1CYP3A4CYP2C19KCNH2
SCHEMBL538933 0.88 MCHR1 (0.73) MCHR1CYP3A4CYP2C19
SCHEMBL539094 0.87 MCHR1 (0.70) MCHR1CYP3A4CYP2C19KCNH2
Hydrochloric Acid SCHEMBL539144 0.87 MCHR1 (0.72) MCHR1CYP3A4CYP2C19
SCHEMBL537233 0.86 MCHR1 (0.77) MCHR1CYP3A4CYP2C19
Hydrochloric Acid SCHEMBL538927 0.86 MCHR1 (0.69) MCHR1CYP3A4CYP2C19KCNH2
SCHEMBL10144451 0.85 MCHR1 (0.72) MCHR1CYP3A4CYP2C19KCNH2
SCHEMBL539062 0.84 MCHR1 (0.90) MCHR1CYP3A4CYP2C19KCNH2
Hydrochloric Acid SCHEMBL539559 0.84 MCHR1 (0.88) MCHR1CYP3A4CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2176251-B1 5-pyridinone substituted indazoles and pharmaceutical compositions thereof ALBANY MOLECULAR RES INC (US) 2012-02-08 EP disclosed
WO-2009015037-A2 5-PYRIDINONE SUBSTITUTED INDAZOLES ALBANY MOLECULAR RESEARCH, INC. (US) 2009-01-29 WO disclosed