SCHEMBL10144674

SCHEMBL10144674

NC(=O)[C@H]1CC[C@@H](NC(=O)c2cccc(F)c2)CC1

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 4/20 0.64
L3MBTL1 Q9Y468 1/20 0.55
KMT2A Q03164 3/20 0.55
MEN1 O00255 2/20 0.55
SMYD3 Q9H7B4 2/20 0.52
CCR3 P51677 1/20 0.52
HTR2B P41595 1/20 0.51
AR P10275 1/20 0.51
HDAC1 Q13547 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
NPC1 O15118 1/20 0.50
ADRA2A P08913 1/20 0.49
MCHR1 Q99705 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1116603 0.90 GRM5 (0.77) GRM5L3MBTL1KMT2AMEN1SMYD3
SCHEMBL23573558 0.84 GRM5 (0.69) GRM5L3MBTL1KMT2AMEN1CCR3
SCHEMBL15962709 0.84 GRM5 (0.69) GRM5L3MBTL1KMT2AMEN1SMYD3
SCHEMBL23573560 0.84 GRM5 (0.69) GRM5L3MBTL1KMT2AMEN1CCR3
SCHEMBL3462086 0.82 GRM5 (0.71) GRM5L3MBTL1KMT2AMEN1CCR3
SCHEMBL13294374 0.82 GRM5 (0.81) GRM5L3MBTL1KMT2AMEN1HTR2B
SCHEMBL12259124 0.82 GRM5 (0.66) GRM5L3MBTL1KMT2AMEN1CCR3
SCHEMBL4403625 0.80 GRM5 (0.68) GRM5L3MBTL1KMT2AMEN1SMYD3
SCHEMBL29639471 0.80 GRM5 (0.68) GRM5L3MBTL1KMT2AMEN1CCR3
SCHEMBL29973192 0.78 KMT2A (0.65) GRM5L3MBTL1KMT2AMEN1CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2404896-A1 CYCLOHEXANE DERIVATIVE HAVING NPY Y5 RECEPTOR ANTAGONISM Shionogi&Co., Ltd. (JP) 2012-01-11 EP disclosed