SCHEMBL10145266

SCHEMBL10145266

CS(=O)(=O)c1cc(OCc2ccccc2)ccc1-c1ccn(-c2ccc3c(cnn3CCN3CCCC3)c2)c(=O)c1

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 20/20 0.73
KCNH2 Q12809 7/20 0.73
CYP3A4 P08684 3/20 0.73
CYP2C19 P33261 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12680001 0.90 MCHR1 (0.78) MCHR1KCNH2CYP3A4CYP2C19
Hydrochloric Acid SCHEMBL539110 0.89 MCHR1 (0.77) MCHR1KCNH2CYP3A4CYP2C19
SCHEMBL539304 0.85 MCHR1 (1.00) MCHR1KCNH2CYP3A4
Hydrochloric Acid SCHEMBL2966575 0.84 MCHR1 (0.98) MCHR1KCNH2CYP3A4
SCHEMBL2962727 0.84 MCHR1 (0.98) MCHR1KCNH2CYP3A4
Hydrochloric Acid SCHEMBL2959155 0.84 MCHR1 (0.96) MCHR1KCNH2CYP3A4
SCHEMBL12340004 0.82 MCHR1 (0.90) MCHR1KCNH2CYP3A4CYP2C19
Hydrochloric Acid SCHEMBL2961905 0.81 MCHR1 (0.88) MCHR1KCNH2CYP3A4CYP2C19
SCHEMBL12340044 0.80 MCHR1 (0.86) MCHR1KCNH2CYP3A4
SCHEMBL12339975 0.80 MCHR1 (0.88) MCHR1KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2176251-B1 5-pyridinone substituted indazoles and pharmaceutical compositions thereof ALBANY MOLECULAR RES INC (US) 2012-02-08 EP disclosed