SCHEMBL10145269

SCHEMBL10145269

O=C(c1cnc(NC2C[C@H]3CC[C@@H]2C3)nc1C(F)(F)F)N1CCS(=O)(=O)CC1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.41
AURKB Q96GD4 1/20 0.41
HRH4 Q9H3N8 4/20 0.40
CXCR4 P61073 1/20 0.38
SCD O00767 1/20 0.38
GABBR2 O75899 7/20 0.38
GABBR1 Q9UBS5 7/20 0.38
CXCR1 P25024 1/20 0.37
CXCR2 P25025 1/20 0.37
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
JAK3 P52333 1/20 0.36
SYK P43405 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10145905 1.00 KDR (0.41) KDRAURKBHRH4CXCR4SCD
SCHEMBL541903 1.00 KDR (0.41) KDRAURKBHRH4CXCR4SCD
SCHEMBL541084 1.00 KDR (0.41) KDRAURKBHRH4CXCR4SCD
SCHEMBL541730 1.00 KDR (0.41) KDRAURKBHRH4CXCR4SCD
SCHEMBL12796694 0.95 CXCR4 (0.39) KDRAURKBHRH4CXCR4SCD
SCHEMBL541902 0.93 KDR (0.41) KDRAURKBHRH4CXCR4SCD
SCHEMBL541731 0.93 KDR (0.41) KDRAURKBHRH4CXCR4SCD
SCHEMBL541729 0.93 KDR (0.41) KDRAURKBHRH4CXCR4SCD
SCHEMBL541904 0.93 KDR (0.41) KDRAURKBHRH4CXCR4SCD
SCHEMBL541083 0.93 KDR (0.41) KDRAURKBHRH4CXCR4SCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415765-A1 PYRIMIDINE COMPOUND Astellas Pharma Inc. (JP) 2012-02-08 EP disclosed