SCHEMBL10148189

SCHEMBL10148189

Bc1cnc(Nc2ccc(C(=O)Cl)cc2)nc1Cl

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
GSK3B P49841 5/20 0.43
GSK3A P49840 4/20 0.43
AURKA O14965 11/20 0.42
JAK2 O60674 4/20 0.41
AURKB Q96GD4 3/20 0.41
NTRK1 P04629 1/20 0.39
LRRK2 Q5S007 1/20 0.39
CSNK2A1 P68400 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2516504 0.83 HDAC3 (0.43) HDAC3HDAC1HDAC2HDAC6GSK3B
SCHEMBL578612 0.83 GSK3B (0.53) HDAC3HDAC1HDAC2HDAC6GSK3B
SCHEMBL10148230 0.83 AURKA (0.48) HDAC3HDAC1HDAC2HDAC6GSK3B
SCHEMBL578690 0.80 GSK3A (0.56) GSK3BGSK3AAURKAJAK2NTRK1
SCHEMBL21725113 0.72 AURKA (0.49) HDAC3HDAC1HDAC2HDAC6AURKA
SCHEMBL14621366 0.71 AURKA (0.59) GSK3BGSK3AAURKAJAK2AURKB
SCHEMBL2523254 0.71 GSK3B (0.54) GSK3BGSK3AAURKAJAK2AURKB
SCHEMBL578613 0.71 GSK3B (0.67) GSK3BGSK3AAURKAJAK2AURKB
SCHEMBL3135192 0.71 SYK (0.56) HDAC3HDAC1HDAC2HDAC6AURKA
SCHEMBL11596462 0.70 MAPK13 (0.52) HDAC3HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2027107-B1 2, 4 -DIAMINO PYRIMIDINES AS CELL CYCLE KINASE INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2012-02-15 EP disclosed