SCHEMBL10175423

SCHEMBL10175423

COC(=O)[C@@H](OC(C)(C)C)c1c(C)nc2c(C)c(-c3ccccc3)nn2c1-c1cc(F)c2c(c1C)CCCO2

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.69
CYP3A4 P08684 2/20 0.34
AKT1 P31749 1/20 0.31
AKT2 P31751 1/20 0.31
PSIP1 O75475 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL463092 1.00 NR1I2 (0.69) NR1I2CYP3A4AKT1AKT2PSIP1
SCHEMBL459580 0.94 NR1I2 (0.68) NR1I2CYP3A4PSIP1
SCHEMBL12091349 0.94 NR1I2 (0.68) NR1I2CYP3A4PSIP1
SCHEMBL462664 0.94 NR1I2 (0.78) NR1I2CYP3A4PSIP1
SCHEMBL461679 0.94 NR1I2 (0.78) NR1I2CYP3A4PSIP1
SCHEMBL461693 0.94 NR1I2 (0.67) NR1I2CYP3A4AKT1AKT2PSIP1
SCHEMBL456824 0.94 NR1I2 (0.67) NR1I2CYP3A4AKT1AKT2PSIP1
SCHEMBL470442 0.94 NR1I2 (0.69) NR1I2CYP3A4PSIP1
SCHEMBL460947 0.92 NR1I2 (0.65) NR1I2CYP3A4PSIP1
SCHEMBL461267 0.92 NR1I2 (0.65) NR1I2CYP3A4PSIP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033735-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-15 WO disclosed