SCHEMBL10180905

SCHEMBL10180905

CCCOc1ccc(CN2CCN(C(=O)c3cc4cc(Oc5ccc(N(C)C(=O)c6ccc(Cl)c(Cl)c6)cn5)ccc4n3C)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 15/20 0.44
MLNR O43193 1/20 0.43
PIK3CA P42336 2/20 0.43
PRKAA2 P54646 2/20 0.43
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL3062043 0.96 STAT3 (0.42) STAT3MLNRPIK3CAPRKAA2
Maleic Acid SCHEMBL3062041 0.96 STAT3 (0.42) STAT3MLNRPIK3CAPRKAA2
Bromide SCHEMBL3046046 0.94 STAT3 (0.49) STAT3MLNR
SCHEMBL3046815 0.92 PIK3CA (0.44) STAT3MLNRPIK3CAPRKAA2
Bromide SCHEMBL3061151 0.91 STAT3 (0.45) STAT3MLNRHRH3
Bromide SCHEMBL10181379 0.91 PIK3CA (0.51) STAT3MLNRPIK3CAPRKAA2HRH3
Bromide SCHEMBL3064130 0.91 STAT3 (0.44) STAT3MLNRPIK3CAPRKAA2HRH3
SCHEMBL10180586 0.90 STAT3 (0.54) STAT3PIK3CAPRKAA2
Maleic Acid SCHEMBL3069658 0.89 STAT3 (0.45) STAT3PIK3CAPRKAA2HRH3
Fumaric Acid SCHEMBL3069662 0.89 STAT3 (0.45) STAT3PIK3CAPRKAA2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2207773-B1 HETEROCYCLIC COMPOUND AND PHARMACEUTICAL COMPOSITION THEREOF OTSUKA PHARMA CO LTD (JP) 2012-07-11 EP disclosed