SCHEMBL10180974

SCHEMBL10180974

CCOc1ccc(CN2CCN(C(=O)c3cc4cc(Oc5ccc(N(C)C(=O)c6ccc(C(F)(F)F)cc6)c(C)n5)ccc4n3C)CC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 19/20 0.51
PIK3CA P42336 1/20 0.48
PRKAA2 P54646 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL10180685 0.99 STAT3 (0.51) STAT3PIK3CAPRKAA2
SCHEMBL3059167 0.93 STAT3 (0.49) STAT3PIK3CAPRKAA2
Bromide SCHEMBL3051528 0.90 STAT3 (0.53) STAT3PIK3CAPRKAA2
SCHEMBL10180482 0.89 STAT3 (0.55) STAT3PIK3CAPRKAA2
Fumaric Acid SCHEMBL3061331 0.86 PIK3CA (0.41) STAT3PIK3CAPRKAA2
Maleic Acid SCHEMBL3061327 0.86 PIK3CA (0.41) STAT3PIK3CAPRKAA2
Maleic Acid SCHEMBL3063405 0.86 STAT3 (0.52) STAT3PIK3CAPRKAA2
Fumaric Acid SCHEMBL3063410 0.86 STAT3 (0.52) STAT3PIK3CAPRKAA2
SCHEMBL3062544 0.85 SCN9A (0.45) STAT3
Bromide SCHEMBL3056975 0.85 STAT3 (0.57) STAT3PIK3CAPRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8551999-B2 Heterocyclic compound and pharmaceutical composition thereof OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2013-10-08 US claimed
EP-2207773-B1 HETEROCYCLIC COMPOUND AND PHARMACEUTICAL COMPOSITION THEREOF OTSUKA PHARMA CO LTD (JP) 2012-07-11 EP claimed