SCHEMBL10181121

SCHEMBL10181121

CCOc1ccc(Cl)cc1C(=O)NCCc1ccc(-c2ccc(OC(=O)O)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DNMT3A Q9Y6K1 1/20 0.56
TP53 P04637 1/20 0.54
HDAC1 Q13547 2/20 0.53
HDAC6 Q9UBN7 2/20 0.53
NLRP3 Q96P20 3/20 0.52
AKR1C3 P42330 1/20 0.50
MAPT P10636 1/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10182210 0.92 DNMT3A (0.54) DNMT3ATP53HDAC1HDAC6NLRP3
SCHEMBL10181010 0.92 DNMT3A (0.54) DNMT3ATP53HDAC1HDAC6NLRP3
SCHEMBL10181758 0.90 DNMT3A (0.53) DNMT3AHDAC1HDAC6NLRP3AKR1C3
SCHEMBL10181170 0.89 DNMT3A (0.52) DNMT3AHDAC1HDAC6NLRP3AKR1C3
SCHEMBL10181246 0.89 DNMT3A (0.53) DNMT3ATP53HDAC1HDAC6NLRP3
SCHEMBL10182293 0.88 DNMT3A (0.50) DNMT3ATP53HDAC1HDAC6NLRP3
SCHEMBL10181905 0.88 DNMT3A (0.58) DNMT3AHDAC1HDAC6NLRP3AKR1C3
SCHEMBL1154293 0.88 DNMT3A (0.58) DNMT3ATP53HDAC1HDAC6NLRP3
SCHEMBL10181772 0.88 DNMT3A (0.52) DNMT3ATP53HDAC1HDAC6NLRP3
SCHEMBL10181767 0.87 DNMT3A (0.51) DNMT3ATP53HDAC1HDAC6NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2215065-B1 CCR10 ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-07-11 EP claimed