SCHEMBL10185525

SCHEMBL10185525

Cc1ccccc1C(C(=O)NC1CCCCC1)N(C(=O)CN1CCN(C(=O)CC(C)C)CC1)c1cccc(F)c1

nearest known ligand 0.81

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 15/20 0.81
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
NPC1 O15118 1/20 0.46
ALDH1A1 P00352 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15118906 0.90 IDH1 (1.00) IDH1MEN1KMT2ANPC1
SCHEMBL10184097 0.89 IDH1 (0.84) IDH1MEN1KMT2ANPC1ALDH1A1
SCHEMBL15119069 0.89 IDH1 (0.84) IDH1MEN1KMT2ANPC1ALDH1A1
SCHEMBL15119072 0.89 IDH1 (0.80) IDH1MEN1KMT2ANPC1
SCHEMBL10185541 0.88 IDH1 (0.86) IDH1MEN1KMT2ANPC1
SCHEMBL10185548 0.87 IDH1 (1.00) IDH1MEN1KMT2ANPC1
SCHEMBL360556 0.87 IDH1 (1.00) IDH1MEN1KMT2ANPC1
SCHEMBL15118975 0.85 IDH1 (0.84) IDH1MEN1KMT2ANPC1
SCHEMBL10185870 0.83 IDH1 (0.81) IDH1MEN1KMT2ANPC1
SCHEMBL15119070 0.83 IDH1 (0.76) IDH1MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012009678-A1 THERAPEUTICALLY ACTIVE COMPOSITIONS AND THEIR METHOD OF USE AGIOS PHARMACEUTICALS, INC. (US) 2012-01-19 WO disclosed