SCHEMBL10187145

SCHEMBL10187145

CCCOc1ccc(N)c(C#N)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.48
ACACB O00763 2/20 0.42
KMT2A Q03164 4/20 0.41
MAOB P27338 2/20 0.41
MEN1 O00255 3/20 0.40
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
HTT P42858 2/20 0.40
KDM4E B2RXH2 1/20 0.40
USP2 O75604 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9072621 0.93 TSHR (0.45) MAPTKMT2AMAOBMEN1CA12
SCHEMBL11790185 0.87 MAPT (0.51) MAPTACACBKMT2AMAOBMEN1
SCHEMBL11796509 0.86 MEN1 (0.54) MAPTKMT2AMAOBMEN1KDM4E
SCHEMBL13876611 0.85 MAOB (0.40) MAOBKDM4EUSP2ALDH1A1CASP1
SCHEMBL13482321 0.84 MAOB (0.56) MAPTACACBKMT2AMAOBCA12
SCHEMBL28017761 0.83 MAOB (0.41) MAPTKMT2AMAOBMEN1KDM4E
SCHEMBL28017766 0.83 MAOB (0.41) MAPTKMT2AMAOBMEN1NPC1
SCHEMBL7356604 0.81 PTGS1 (0.45) MAPTACACBKMT2AMAOBCA12
SCHEMBL175022 0.80 ACACB (0.42) MAPTACACBKMT2AMAOBCA12
SCHEMBL1697625 0.80 MAOB (0.45) MAPTACACBKMT2AMAOBCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012001107-A1 PIPERIDINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF METABOLIC DISORDERS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-05 WO disclosed