SCHEMBL10187282

SCHEMBL10187282

Nc1ccnc(N2CC3CCCC3C2)n1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.49
KDM1A O60341 1/20 0.43
SMPD3 Q9NY59 1/20 0.40
ACACB O00763 3/20 0.39
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
OGA O60502 1/20 0.36
PDE10A Q9Y233 1/20 0.35
HCRTR2 O43614 8/20 0.34
HCRTR1 O43613 7/20 0.34
HRH3 Q9Y5N1 1/20 0.34
CDC7 O00311 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30075754 0.84 KDM1A (0.41) DYRK1AKDM1AMKNK1MKNK2OGA
SCHEMBL24969806 0.84 KDM1A (0.41) DYRK1AKDM1AMKNK1MKNK2OGA
SCHEMBL23579347 0.82 KDM1A (0.40) DYRK1AKDM1AMKNK1MKNK2OGA
SCHEMBL23593411 0.82 KDM1A (0.40) DYRK1AKDM1AMKNK1MKNK2OGA
SCHEMBL30556681 0.80 HCRTR2 (0.49) DYRK1AACACBHCRTR2HCRTR1
SCHEMBL23593409 0.80 KDM1A (0.46) DYRK1AKDM1ASMPD3MKNK1MKNK2
SCHEMBL29959199 0.79 KDM1A (0.42) DYRK1AKDM1AMKNK1MKNK2OGA
SCHEMBL23579408 0.79 KDM1A (0.42) DYRK1AKDM1AMKNK1MKNK2OGA
SCHEMBL4949146 0.79 MTOR (0.45) KDM1AACACBMKNK1MKNK2OGA
SCHEMBL10187275 0.77 KDM1A (0.48) DYRK1AKDM1AMKNK1MKNK2OGA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012001107-A1 PIPERIDINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF METABOLIC DISORDERS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-05 WO disclosed