SCHEMBL10187341

SCHEMBL10187341

CC(C)(C)OC(=O)n1c(B(O)O)cc2cc(N)ccc21

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 14/20 0.41
NR1H3 Q13133 3/20 0.38
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
CHEK1 O14757 1/20 0.36
AURKA O14965 1/20 0.36
DAPK3 O43293 1/20 0.36
CSNK1A1 P48729 1/20 0.36
GSK3A P49840 1/20 0.36
LIMK1 P53667 1/20 0.36
IKBKE Q14164 1/20 0.36
MAPK14 Q16539 1/20 0.36
TAOK1 Q7L7X3 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
BRPF1 P55201 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL593975 0.85 NR1H2 (0.44) NR1H2NR1H3CA12CA9GABRG2
SCHEMBL29957250 0.85 NR1H2 (0.44) NR1H2NR1H3CA12CA9GABRG2
SCHEMBL17690271 0.85 ESR2 (0.40) NR1H2NR1H3CA12CA9GABRG2
SCHEMBL29643728 0.84 NR1H2 (0.45) NR1H2NR1H3CA12CA9GABRG2
SCHEMBL2930214 0.84 NR1H2 (0.39) NR1H2NR1H3CA12CA9GABRG2
SCHEMBL7921587 0.84 CCNB2 (0.41) NR1H2NR1H3CA12CA9GABRG2
SCHEMBL29955454 0.84 NR1H2 (0.39) NR1H2NR1H3CA12CA9GABRG2
SCHEMBL31140070 0.84 CCNB2 (0.41) NR1H2NR1H3CA12CA9GABRG2
SCHEMBL594560 0.84 NR1H2 (0.45) NR1H2NR1H3CA12CA9GABRG2
SCHEMBL29955030 0.83 NR1H2 (0.46) NR1H2CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012001107-A1 PIPERIDINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF METABOLIC DISORDERS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-05 WO disclosed