SCHEMBL10187464

SCHEMBL10187464

CCOc1cccc(-c2cc([C@]3(C)CC(=O)N(C)C(=N)N3)ccn2)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 10/20 0.39
CTSD P07339 1/20 0.39
MAPT P10636 3/20 0.37
GAA P10253 2/20 0.37
KDM4E B2RXH2 1/20 0.37
THRB P10828 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TP53 P04637 1/20 0.35
FYN P06241 1/20 0.35
MAPKAPK2 P49137 1/20 0.34
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34
BUB1 O43683 1/20 0.33
MGAT2 Q10469 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7543537 0.90 BACE1 (0.48) BACE1CTSDMAPKAPK2
SCHEMBL4549225 0.88 BACE1 (0.36) BACE1MAPKAPK2
SCHEMBL7600700 0.87 SCN9A (0.42) BACE1CTSD
SCHEMBL8437193 0.85 CYP2A6 (0.36) BACE1
SCHEMBL13407696 0.84 MAPKAPK2 (0.39) BACE1MEN1KMT2AMAPKAPK2
SCHEMBL7539812 0.84 MAPKAPK2 (0.39) BACE1MEN1KMT2AMAPKAPK2
SCHEMBL8433127 0.84 MAPKAPK2 (0.39) BACE1KDM4EHSD17B10FYNMAPKAPK2
SCHEMBL7544553 0.84 BACE1 (0.40) BACE1CTSDMAPTGAAKDM4E
SCHEMBL7538440 0.82 BACE1 (0.49) BACE1CTSD
SCHEMBL4549230 0.82 BACE1 (0.39) BACE1CTSDBUB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8168641-B2 Aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-01 US disclosed