SCHEMBL10194503

SCHEMBL10194503

Cn1c(C(N)=O)c(N)c2c(-c3ccc(CCCO)cc3)c(C#N)c(SCc3cccc(C(N)=O)c3)nc21

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 20/20 0.55
ADORA2B P29275 4/20 0.49
ADORA2A P29274 6/20 0.48
ADORA3 P0DMS8 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10194477 0.96 ADORA1 (0.53) ADORA1ADORA2BADORA2AADORA3
SCHEMBL382496 0.89 ADORA1 (0.58) ADORA1ADORA2BADORA2AADORA3
SCHEMBL10194562 0.88 ADORA1 (0.51) ADORA1ADORA2BADORA2AADORA3
SCHEMBL8030215 0.85 ADORA1 (0.54) ADORA1ADORA2BADORA2AADORA3
SCHEMBL8038927 0.85 ADORA1 (0.46) ADORA1ADORA2BADORA2AADORA3
SCHEMBL382755 0.83 ADORA1 (0.55) ADORA1ADORA2BADORA2AADORA3
SCHEMBL8034138 0.81 ADORA1 (0.54) ADORA1
SCHEMBL8032331 0.78 ADORA1 (0.55) ADORA1ADORA2BADORA2AADORA3
SCHEMBL8036775 0.78 ADORA1 (0.55) ADORA1ADORA2BADORA2AADORA3
SCHEMBL10194487 0.77 ADORA1 (0.77) ADORA1ADORA2BADORA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2235011-B1 SUBSTITUTED PYRROLO[2, 3-B]AND PYRAZOLO[3, 4-B]PYRIDINES FOR USE AS ADENOSINE RECEPTOR LIGANDS Bayer Pharma AG (DE) 2012-01-25 EP disclosed