SCHEMBL10197546

SCHEMBL10197546

O=C(OCc1ccccc1)N1CC(O)(C(=O)O)C1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.56
MEN1 O00255 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
SMN1; SMN2 Q16637 4/20 0.55
NPC1 O15118 4/20 0.55
RAB9A P51151 4/20 0.55
CYP2C19 P33261 1/20 0.52
L3MBTL1 Q9Y468 2/20 0.47
HTR2C P28335 2/20 0.47
P2RX4 Q99571 2/20 0.47
ALDH1A1 P00352 3/20 0.46
MAPK1 P28482 2/20 0.46
GAA P10253 1/20 0.46
P2RX1 P51575 1/20 0.46
P2RX3 P56373 1/20 0.46
SLC6A2 P23975 1/20 0.45
SLC6A3 Q01959 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
HTR1A P08908 1/20 0.44
ADRA2A P08913 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11545254 0.90 MEN1 (0.56) KMT2AMEN1NPSR1SMN1; SMN2NPC1
SCHEMBL6827246 0.85 MEN1 (0.61) KMT2AMEN1NPSR1SMN1; SMN2NPC1
SCHEMBL2673587 0.84 KMT2A (0.56) KMT2AMEN1NPSR1SMN1; SMN2NPC1
SCHEMBL3919116 0.83 MEN1 (0.55) KMT2AMEN1NPSR1SMN1; SMN2NPC1
SCHEMBL11613000 0.83 MEN1 (0.55) KMT2AMEN1NPSR1SMN1; SMN2NPC1
SCHEMBL22075574 0.83 KMT2A (0.55) KMT2AMEN1NPSR1SMN1; SMN2NPC1
SCHEMBL29220951 0.82 MEN1 (0.54) KMT2AMEN1NPSR1SMN1; SMN2NPC1
SCHEMBL3151804 0.82 KMT2A (0.54) KMT2AMEN1NPSR1SMN1; SMN2NPC1
SCHEMBL18204368 0.82 MEN1 (0.54) KMT2AMEN1NPSR1SMN1; SMN2NPC1
SCHEMBL9217126 0.81 KMT2A (0.56) KMT2AMEN1NPSR1SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116789636-A Bifunctional compound, preparation method, pharmaceutical composition and application thereof 北京康辰药业股份有限公司 2023-09-22 CN disclosed
WO-2011044538-A9 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2012-01-05 WO disclosed
WO-2011044538-A1 ANTIBACTERIAL AMINOGLYCOSIDE ANALOGS ACHAOGEN, INC. (US) 2011-04-14 WO disclosed
EP-0001280-B1 1-N-ACYLATED-4-O-GLYCOSYL-6-O-GLYCOSYL-1,3-DIAMINOCYCLITOL DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SHIONOGI & CO., LTD. (JP) 1981-11-25 EP disclosed
US-4199570-A AZETIDINE, PYRROLIDINE, OR PIPERIDINE SHIONOGI & CO., LTD. (JP) 1980-04-22 US disclosed
EP-0001280-A2 1-N-acylated-4-O-glycosyl-6-O-glycosyl-1,3-diaminocyclitol derivatives, process for their preparation and pharmaceutical compositions containing them SHIONOGI & CO., LTD. (JP) 1979-04-04 EP disclosed