SCHEMBL10210895

SCHEMBL10210895

Cc1noc(-c2ccccc2)c1CN1CCCCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MAPT P10636 2/20 0.47
RAB9A P51151 2/20 0.45
KMT2A Q03164 2/20 0.45
ATM Q13315 1/20 0.45
HCRTR1 O43613 1/20 0.45
HCRTR2 O43614 1/20 0.45
SIGMAR1 Q99720 1/20 0.43
NPC1 O15118 1/20 0.43
SLC6A9 P48067 1/20 0.43
GAA P10253 2/20 0.42
BRD4 O60885 1/20 0.41
LMNA P02545 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
GRIN2B Q13224 4/20 0.41
CYP2D6 P10635 2/20 0.41
CYP1A2 P05177 1/20 0.41
GRIN1 Q05586 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15084374 0.83 HRH3 (0.45) ALDH1A1MAPTRAB9AKMT2AHCRTR1
SCHEMBL10212867 0.82 HCRTR1 (0.42) ALDH1A1SMN1; SMN2MAPTKMT2AATM
SCHEMBL15081973 0.81 HCRTR1 (0.39) ALDH1A1SMN1; SMN2MAPTATMHCRTR1
SCHEMBL10210892 0.77 KMT2A (0.51) ALDH1A1SMN1; SMN2RAB9AKMT2AATM
SCHEMBL8976521 0.76 BRD4 (0.48) ALDH1A1SMN1; SMN2MAPTKMT2AHCRTR1
SCHEMBL4655 0.76 SLC18A3 (0.45) ALDH1A1SMN1; SMN2KMT2AGAALMNA
SCHEMBL31010210 0.75 BRD4 (0.49) ALDH1A1SMN1; SMN2RAB9ASIGMAR1NPC1
Bicarbonate SCHEMBL18167217 0.74 OGA (0.45) ALDH1A1SMN1; SMN2RAB9AKMT2ASIGMAR1
SCHEMBL6261211 0.74 HCRTR1 (0.39) ALDH1A1SMN1; SMN2MAPTHCRTR1HCRTR2
SCHEMBL2413945 0.73 BRD4 (0.46) ALDH1A1SMN1; SMN2MAPTKMT2ASLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012036997-A1 FUSED PYRAZOLE DERIVATIVES AS NOVEL ERK INHIBITORS SCHERING CORPORATION (US) 2012-03-22 WO disclosed