SCHEMBL1021269

SCHEMBL1021269

CCCCN(C(=O)O)C(C)CN

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.35
CA1 P00915 2/20 0.35
CA9 Q16790 2/20 0.35
EPHX2 P34913 1/20 0.35
GPR84 Q9NQS5 3/20 0.34
FFAR1 O14842 1/20 0.34
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33
MMP3 P08254 1/20 0.33
MMP8 P22894 1/20 0.33
DNM1 Q05193 1/20 0.33
ACE2 Q9BYF1 1/20 0.32
ALOX15 P16050 1/20 0.31
CA2 P00918 1/20 0.31
MAPK1 P28482 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
AKR1B1 P15121 1/20 0.31
KDM5A P29375 2/20 0.31
KDM4C Q9H3R0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11355835 0.93 EPHX2 (0.42) EPHX2GPR84FFAR1DNM1ACE2
SCHEMBL16197622 0.82 CA1 (0.36) CA12CA1CA9EPHX2GPR84
SCHEMBL28783746 0.82 CHRM1 (0.37) CA12CA1CA9EPHX2GPR84
SCHEMBL15589936 0.82 CA1 (0.36) CA12CA1CA9EPHX2GPR84
SCHEMBL3669268 0.81 CA1 (0.35) CA12CA1CA9EPHX2GPR84
SCHEMBL20186794 0.79 GABRR1 (0.33)
SCHEMBL20186754 0.79 GABRR1 (0.33)
SCHEMBL1758802 0.79 EPHX2 (0.45) CA12CA1CA9EPHX2GPR84
SCHEMBL20186756 0.79 GABRR1 (0.33)
SCHEMBL10529104 0.76 CA12 (0.42) CA12CA1CA9EPHX2GPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274300-A2 NOVEL HETEROCYCLIC COMPOUNDS AND USES THEROF Novartis AG (CH) 2011-01-19 EP disclosed
WO-2009115572-A2 NOVEL HETEROCYCLIC COMPOUNDS AND USES THEROF NOVARTIS AG (CH) 2009-09-24 WO disclosed