SCHEMBL10219342

SCHEMBL10219342

Cn1nc(C(N)=O)c2c1-c1nc(Oc3ccc(I)cc3Br)ncc1CC2

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 16/20 0.55
CCNA2 P20248 18/20 0.54
CDK2 P24941 18/20 0.54
CCNA1 P78396 16/20 0.54
AURKA O14965 10/20 0.53
PLK3 Q9H4B4 9/20 0.53
PLK2 Q9NYY3 9/20 0.53
TTK P33981 4/20 0.53
CDK4 P11802 3/20 0.53
CCND3 P30281 3/20 0.53
CDK6 Q00534 3/20 0.53
RPS6KA4 O75676 1/20 0.51
CDK1 P06493 1/20 0.51
KIT P10721 1/20 0.51
IMPDH2 P12268 1/20 0.51
CCNB1 P14635 1/20 0.51
CSNK2A2 P19784 1/20 0.51
CCNE1 P24864 1/20 0.51
FLT4 P35916 1/20 0.51
CSNK1D P48730 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11025830 0.86 PLK1 (0.65) PLK1CCNA2CDK2CCNA1AURKA
SCHEMBL10218678 0.85 CCNA2 (0.59) PLK1CCNA2CDK2CCNA1AURKA
Trifluoroacetic Acid SCHEMBL11023473 0.82 PLK1 (0.63) PLK1CCNA2CDK2CCNA1AURKA
SCHEMBL9940866 0.80 CCNA2 (0.61) PLK1CCNA2CDK2CCNA1AURKA
SCHEMBL9940913 0.80 CCNA2 (0.65) PLK1CCNA2CDK2CCNA1AURKA
SCHEMBL9940668 0.80 CCNA2 (0.65) PLK1CCNA2CDK2CCNA1AURKA
SCHEMBL9940794 0.79 CCNA2 (0.69) PLK1CCNA2CDK2CCNA1AURKA
SCHEMBL9940400 0.78 CCNA2 (0.64) PLK1CCNA2CDK2CCNA1AURKA
SCHEMBL9940837 0.78 CCNA2 (0.60) PLK1CCNA2CDK2CCNA1AURKA
SCHEMBL10220009 0.78 PLK1 (0.65) PLK1CCNA2CDK2CCNA1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012080990-A1 SUBSTITUTED PYRAZOLO-QUINAZOLINE DERIVATIVES AS KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2012-06-21 WO disclosed