SCHEMBL10227136

SCHEMBL10227136

CCc1cccc2nc(C)[nH]c(=O)c12

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.68
TYMS P04818 9/20 0.54
ELANE P08246 5/20 0.54
TNKS2 Q9H2K2 1/20 0.53
BMPR1B O00238 1/20 0.46
RAF1 P04049 1/20 0.46
BRAF P15056 1/20 0.46
BMPR1A P36894 1/20 0.46
ACVR1B P36896 1/20 0.46
TGFBR1 P36897 1/20 0.46
ACVRL1 P37023 1/20 0.46
ACVR1 Q04771 1/20 0.46
KDM4E B2RXH2 1/20 0.45
NPC1 O15118 1/20 0.45
USP2 O75604 1/20 0.45
ALDH1A1 P00352 1/20 0.45
GLA P06280 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30838794 0.81 PARP1 (1.00) PARP1TYMSELANETNKS2BMPR1B
SCHEMBL9259148 0.81 PARP1 (1.00) PARP1TYMSELANETNKS2BMPR1B
SCHEMBL30704850 0.78 PARP1 (1.00) PARP1TYMSTNKS2BMPR1BRAF1
SCHEMBL2659299 0.78 PARP1 (1.00) PARP1TYMSTNKS2BMPR1BRAF1
SCHEMBL29964360 0.78 PARP1 (1.00) PARP1TYMSTNKS2BMPR1BRAF1
SCHEMBL12169915 0.78 PARP1 (1.00) PARP1TYMSTNKS2BMPR1BRAF1
SCHEMBL328456 0.78 PARP1 (0.70) PARP1TYMSTNKS2BMPR1BRAF1
SCHEMBL29442253 0.78 PARP1 (0.70) PARP1TYMSTNKS2BMPR1BRAF1
SCHEMBL20169191 0.77 PARP1 (0.46) PARP1TYMSELANETNKS2KDM4E
SCHEMBL19936540 0.75 PARP1 (0.66) PARP1TYMSELANETNKS2BMPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8518970-B2 Compounds and methods of use ABBVIE INC. (US) 2013-08-27 US disclosed
US-8114893-B2 Compounds and methods of use GENENTECH, INC. (US) 2012-02-14 US disclosed