SCHEMBL10230604

SCHEMBL10230604

CC(N)c1cccc(-c2cc(-c3nc(-c4ccc(=O)n(C(C)C)c4)cnc3N)on2)c1

nearest known ligand 0.73

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ATR Q13535 19/20 0.73
ATM Q13315 4/20 0.56
PRKDC P78527 2/20 0.56
GSK3B P49841 1/20 0.53
BMPR1B O00238 1/20 0.51
BMPR1A P36894 1/20 0.51
TGFBR1 P36897 1/20 0.51
ACVRL1 P37023 1/20 0.51
ACVR1 Q04771 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10228677 0.92 ATR (0.74) ATRATMPRKDCGSK3B
SCHEMBL10230586 0.92 ATR (0.63) ATRATMPRKDCGSK3B
SCHEMBL18774332 0.92 ATR (0.65) ATRATMPRKDCGSK3B
SCHEMBL506688 0.91 ATR (0.62) ATRATMPRKDCGSK3BBMPR1B
SCHEMBL10231314 0.87 ATR (0.65) ATRATMPRKDCGSK3B
SCHEMBL10230626 0.86 ATR (0.75) ATRATMPRKDCGSK3B
SCHEMBL506418 0.86 ATR (0.81) ATRATMGSK3BBMPR1BBMPR1A
SCHEMBL10177710 0.85 ATR (0.53) ATRATMPRKDCBMPR1BBMPR1A
SCHEMBL506116 0.84 ATR (1.00) ATRATMPRKDCGSK3B
SCHEMBL10229894 0.84 ATR (0.57) ATRATMPRKDCGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9630956-B2 Compounds useful as inhibitors of ATR kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2017-04-25 US disclosed
US-20120027874-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-02-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120027874-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE ATR, CHEK1, CHEK2 ATR 1/4885ATM 32/4885PRKDC 26/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.