SCHEMBL10239277

SCHEMBL10239277

C[C@@H]1COCCN1Cc1nnnn1-c1ccc(N)c(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
LMNA P02545 2/20 0.39
THRB P10828 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PIK3CA P42336 6/20 0.38
MTOR P42345 5/20 0.38
CNR2 P34972 1/20 0.37
NOTUM Q6P988 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
POLB P06746 1/20 0.35
HTT P42858 1/20 0.35
GRM2 Q14416 1/20 0.35
FGFR1 P11362 1/20 0.34
FGFR2 P21802 1/20 0.34
FGFR3 P22607 1/20 0.34
PIK3C3 Q8NEB9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15169040 0.86 AR (0.40) ALDH1A1MEN1KMT2ACYP1A2CYP2C19
SCHEMBL15179487 0.84 CYP1A2 (0.46) ALDH1A1MEN1KMT2ACYP1A2CYP2C19
SCHEMBL324081 0.84 CYP1A2 (0.46) ALDH1A1MEN1KMT2ACYP1A2CYP2C19
Hydrochloric Acid SCHEMBL15168429 0.83 CYP1A2 (0.46) ALDH1A1MEN1KMT2ACYP1A2CYP2C19
Hydrochloric Acid SCHEMBL15168048 0.83 CYP1A2 (0.46) ALDH1A1MEN1KMT2ACYP1A2CYP2C19
SCHEMBL325111 0.82 CNR2 (0.49) ALDH1A1MEN1KMT2ACYP1A2CYP2C19
Hydrochloric Acid SCHEMBL15168744 0.82 CNR2 (0.49) ALDH1A1MEN1KMT2ACYP1A2CYP2C19
SCHEMBL16199555 0.81 CYP1A2 (0.37) ALDH1A1MEN1KMT2ACYP1A2CYP2C19
SCHEMBL16199558 0.75 PRMT1 (0.45) ALDH1A1MEN1KMT2ACYP1A2CYP2C19
SCHEMBL10239578 0.75 PRMT1 (0.45) ALDH1A1MEN1KMT2ACYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012004604-A1 TETRAZOLE COMPOUNDS AS CALCIUM CHANNEL BLOCKERS Convergence Pharmaceuticals Limited (GB) 2012-01-12 WO disclosed