SCHEMBL10246578

SCHEMBL10246578

Nc1ccc(C(=O)N2CCc3nc(COc4cccc(F)c4)oc3C2)cc1F

nearest known ligand 0.85

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 18/20 0.85
CYP2C9 P11712 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL254053 0.93 GRM5 (0.85) GRM5CYP2C9
SCHEMBL10246588 0.92 GRM5 (0.72) GRM5CYP2C9
SCHEMBL156876 0.92 GRM5 (1.00) GRM5
SCHEMBL158401 0.90 GRM5 (1.00) GRM5
SCHEMBL155829 0.89 GRM5 (1.00) GRM5
SCHEMBL173473 0.88 GRM5 (0.81) GRM5
SCHEMBL159568 0.88 GRM5 (1.00) GRM5CYP2C9
SCHEMBL158791 0.88 GRM5 (1.00) GRM5CYP2C9
SCHEMBL170395 0.86 GRM5 (0.81) GRM5
SCHEMBL157534 0.86 GRM5 (0.91) GRM5CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031024-A1 BICYCLIC OXAZOLE AND THIAZOLE COMPOUNDS AND THEIR USE AS ALLOSTERIC MODULATORS OF MGLUR5 RECEPTORS VANDERBILT UNIVERSITY (US) 2012-03-08 WO disclosed