SCHEMBL10265152

SCHEMBL10265152

O=CCCN1CCC2(CC1)COc1cc(OCc3cc(-c4ccccc4)cs3)ccc12

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
S1PR5 Q9H228 20/20 0.56
S1PR1 P21453 12/20 0.53
S1PR3 Q99500 4/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10266087 0.89 S1PR5 (0.51) S1PR5S1PR1S1PR3
SCHEMBL326726 0.88 S1PR5 (0.74) S1PR5S1PR1S1PR3
SCHEMBL10265154 0.85 S1PR5 (0.53) S1PR5S1PR1S1PR3
SCHEMBL10265033 0.84 S1PR5 (0.50) S1PR5S1PR1S1PR3
SCHEMBL326261 0.83 S1PR5 (0.60) S1PR5S1PR1S1PR3
SCHEMBL10268790 0.82 S1PR5 (0.50) S1PR5S1PR1S1PR3
SCHEMBL10266038 0.80 S1PR5 (0.61) S1PR5S1PR1S1PR3
SCHEMBL10265832 0.79 S1PR5 (0.67) S1PR5S1PR1S1PR3
SCHEMBL325892 0.79 S1PR5 (0.68) S1PR5S1PR1S1PR3
SCHEMBL10266036 0.78 S1PR5 (0.76) S1PR5S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012004378-A1 SPIRO-CYCLIC AMINE DERIVATIVES AS S1P MODULATORS ABBOTT HEALTHCARE PRODUCTS B.V. (NL) 2012-01-12 WO disclosed