SCHEMBL10265388

SCHEMBL10265388

COC[C@H](Nc1cc(C(C)(C)C)sc1C(=O)OC)C(=O)N1CCCC1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 18/20 0.48
MAPK14 Q16539 7/20 0.47
MAPK13 O15264 1/20 0.46
MAPK12 P53778 1/20 0.46
MAPK11 Q15759 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15130678 0.83 NR1I2 (0.33) RAF1MAPK14MAPK13MAPK12MAPK11
SCHEMBL10264602 0.81 RAF1 (0.46) RAF1MAPK14MAPK13MAPK12MAPK11
SCHEMBL10264742 0.81 RAF1 (0.46) RAF1MAPK14MAPK13MAPK12MAPK11
SCHEMBL10264610 0.80 RAF1 (0.48) RAF1MAPK14MAPK13MAPK12MAPK11
SCHEMBL14726870 0.76 RAF1 (0.56) RAF1MAPK14MAPK13MAPK12MAPK11
SCHEMBL10268632 0.75 RAF1 (0.51) RAF1MAPK14MAPK13MAPK12MAPK11
SCHEMBL326054 0.75 CYP2E1 (0.41) RAF1
SCHEMBL326053 0.75 CYP2E1 (0.41) RAF1
SCHEMBL10265817 0.72 RAF1 (0.48) RAF1MAPK14MAPK13MAPK12MAPK11
SCHEMBL10264995 0.72 MAPK14 (0.50) RAF1MAPK14MAPK13MAPK12MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006055-A2 COMPOUNDS AND METHODS FOR THE TREATMENT OR PREVENTION OF FLAVIVIRUS INFECTIONS VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-01-12 WO disclosed