SCHEMBL10270150

SCHEMBL10270150

Cc1nc(Cl)cc2nccn12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.35
CLK4 Q9HAZ1 2/20 0.33
CDK8 P49336 2/20 0.33
ROCK1 Q13464 2/20 0.33
FLT1 P17948 1/20 0.33
CDK9 P50750 1/20 0.33
LIMK1 P53667 1/20 0.33
LMNA P02545 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PDE10A Q9Y233 1/20 0.32
DPP4 P27487 1/20 0.31
PDE2A O00408 1/20 0.30
MAP4K2 Q12851 2/20 0.30
AURKB Q96GD4 2/20 0.30
DYRK1B Q9Y463 2/20 0.30
ABL1 P00519 1/20 0.30
PDGFRA P16234 1/20 0.30
CSNK1A1 P48729 1/20 0.30
CDK7 P50613 1/20 0.30
BTK Q06187 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13153127 0.80 PDE2A (0.39) ADORA2ACLK4CDK8ROCK1FLT1
SCHEMBL2571757 0.80 PDE10A (0.33) ADORA2ACDK8ROCK1PDE10AMAP4K2
SCHEMBL2571208 0.77 PDE10A (0.32) CDK8ROCK1PDE10AMAP4K2AURKB
SCHEMBL24174399 0.77 KDM4E (0.41) CLK4CDK8ROCK1FLT1CDK9
SCHEMBL16629908 0.77 DYRK1A (0.40) ADORA2ACLK4CDK8ROCK1FLT1
SCHEMBL27360956 0.77 ABL1 (0.35) ADORA2AABL1KDR
SCHEMBL3607789 0.77 CYP1A2 (0.36) ADORA2A
SCHEMBL10830372 0.77 ADORA2A (0.33) ADORA2ACLK4CDK8ROCK1FLT1
Hydrochloric Acid SCHEMBL2573564 0.75 CYP1A2 (0.35)
SCHEMBL28873688 0.73 ADORA2A (0.37) ADORA2ACLK4CDK8ROCK1FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3356345-B1 HETEROARYL DERIVATIVES AS SEPIAPTERIN REDUCTASE INHIBITORS MAX PLANCK GESELLSCHAFT (DE) 2023-11-08 EP disclosed
EP-2137188-B1 SUBSTITUTED IMIDAZOPYRIMIDINES AND TRIAZOLOPYRIMIDINES Bayer Pharma AG (DE) 2012-06-06 EP disclosed
WO-2008113469-A2 SUBSTITUTED IMIDAZOPYRIMIDINES AND TRIAZOLOPYRIMIDINES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-09-25 WO disclosed