SCHEMBL10270599

SCHEMBL10270599

COC1CCC(C)(C2(c3cc(NC(=O)c4oc5cc(Cl)ccc5c4C)ccc3C)N=C(C)C(N)=N2)CC1

nearest known ligand 0.78

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 18/20 0.78
APP P05067 15/20 0.78
THRB P10828 1/20 0.38
PKM P14618 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18927185 0.88 BACE1 (1.00) BACE1APP
SCHEMBL9948882 0.88 BACE1 (1.00) BACE1APP
SCHEMBL9948883 0.88 BACE1 (1.00) BACE1APP
SCHEMBL21654465 0.87 BACE1 (0.70) BACE1APPTHRBPKMRXFP1
SCHEMBL9948594 0.82 BACE1 (0.89) BACE1APP
SCHEMBL19566705 0.81 BACE1 (0.77) BACE1APP
SCHEMBL18926487 0.70 BACE1 (0.65) BACE1APP
SCHEMBL9948169 0.70 BACE1 (1.00) BACE1APP
SCHEMBL9948016 0.70 BACE1 (1.00) BACE1APP
SCHEMBL18926458 0.69 BACE1 (0.68) BACE1APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087237-A1 COMPOUNDS AND THEIR USE AS BACE INHIBITORS ASTRAZENECA AB (SE) 2012-06-28 WO disclosed