SCHEMBL10280754

SCHEMBL10280754

O=C(Nc1cc2cccnc2cc1OC1CC[C@H](O)C1)c1csc2cncnc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 20/20 1.00
IRAK1 P51617 9/20 1.00
SYK P43405 7/20 1.00
AURKA O14965 1/20 0.75
MAP3K7 O43318 1/20 0.75
FLT3 P36888 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19265933 1.00 IRAK4 (1.00) IRAK4IRAK1SYKAURKAMAP3K7
SCHEMBL10254038 1.00 IRAK4 (1.00) IRAK4IRAK1SYKAURKAMAP3K7
SCHEMBL10254407 1.00 IRAK4 (1.00) IRAK4IRAK1SYKAURKAMAP3K7
Hydrochloric Acid SCHEMBL359133 0.99 IRAK4 (0.98) IRAK4IRAK1SYKAURKAMAP3K7
Hydrochloric Acid SCHEMBL358125 0.99 IRAK4 (0.98) IRAK4IRAK1SYKAURKAMAP3K7
Hydrochloric Acid SCHEMBL358360 0.99 IRAK4 (0.98) IRAK4IRAK1SYKAURKAMAP3K7
SCHEMBL10258448 0.97 IRAK4 (1.00) IRAK4IRAK1SYKAURKAMAP3K7
SCHEMBL358424 0.97 IRAK4 (1.00) IRAK4IRAK1SYKAURKAMAP3K7
SCHEMBL10253920 0.97 IRAK4 (1.00) IRAK4IRAK1SYKAURKAMAP3K7
Hydrochloric Acid SCHEMBL358979 0.96 IRAK4 (0.98) IRAK4IRAK1SYKAURKAMAP3K7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007375-A1 PYRAZOLO [1, 5A] PYRIMIDINE AND THIENO [3, 2B] PYRIMIDINE DERIVATIVES AS IRAK4 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed